Risultati ricerca pubblicazioni

Leveraging the cruzain S3 subsite to increase affinity for reversible covalent inhibitors

pubblicato su: BIOORGANIC CHEMISTRY - 2018

Cianni Lorenzo, Sartori Geraldo, Rosini Fabiana, De Vita Daniela, Pires Gabriel, Lopes Bianca Rebelo, Leitão Andrei, Burtoloso Antonio C B, Montanari Carlos A

Oregonin from Alnus incana bark affects DNA methyltransferases expression and mitochondrial DNA copies in mouse embryonic fibroblasts

pubblicato su: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY - 2018

Krasilnikova Jelena, Lauberte Liga, Stoyanova Elena, Abadjieva Desislava, Chervenkov Mihail, Mori Mattia, De Paolis Elisa, Mladenova Vanya, Telysheva Galina, Botta Bruno, Kistanova Elena

4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis

pubblicato su: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY - 2019

Secci Daniela, Carradori Simone, Petzer Anél, Guglielmi Paolo, D’Ascenzio Melissa, Chimenti Paola, Bagetta Donatella, Alcaro Stefano, Zengin Gokhan, Petzer Jacobus P., Ortuso Francesco

Synthesis and characterisation of a new benzamide-containing nitrobenzoxadiazole as a GSTP1-1 inhibitor endowed with high stability to metabolic hydrolysis

pubblicato su: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY - 2019

Di Paolo V., Fulci C., Rotili D., Sciarretta F., Lucidi A., Morozzo della Rocca B., De Luca A., Rosato A., Quintieri L., Caccuri A. M.

Hydrogen bonding as a clustering agent in protic ionic liquids: like-charge vs opposite-charge dimer formation

pubblicato su: ACS OMEGA - 2018

Le Donne Andrea, Adenusi Henry, Porcelli Francesco, Bodo Enrico

Synthesis, biological evaluation and molecular modeling studies on novel quinonoid inhibitors of CDC25 phosphatases

pubblicato su: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY - 2017

Evain Bana Emilie, Schiavo Lucie, Bour Christophe, Lanfranchi Don Antoine, Berardozzi Simone, Ghirga Francesca, Bagrel Denyse, Botta Bruno, Hanquet Gilles, Mori Mattia

The influence of pH on the scleroglucan and scleroglucan/borax systems

pubblicato su: MOLECULES - 2017

Mazzuca Claudia, Bocchinfuso Gianfranco, Palleschi Antonio, Conflitti Paolo, Grassi Mario, Di Meo Chiara, Alhaique Franco, Coviello Tommasina

Analysis of imidazoles and triazoles in biological samples after MicroExtraction by packed sorbent

pubblicato su: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY - 2017

Campestre Cristina, Locatelli Marcello, Guglielmi Paolo, De Luca Elisa, Bellagamba Giuseppe, Menta Sergio, Zengin Gokhan, Celia Christian, Di Marzio Luisa, Carradori Simone

Efficient synthesis and first regioselective C-6 direct arylation of imidazo[2,1-c][1,2,4]triazine scaffold and their evaluation in H2O2-induced oxidative stress

pubblicato su: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 2018

Loubidi Mohammed, Jouha Jabrane, Tber Zahira, Khouili Mostafa, Suzenet Franck, Akssira Mohamed, Erdogan Mümin Alper, Köse Fadime Aydın, Dagcı Taner, Armagan Güliz, Saso Luciano, Guillaumet Gérald

9-(4'-dimethylaminophenyl)-2,6,7-trihydroxy-xanthene-3-one is a potentially novel antiplatelet drug which antagonizes the effect of thromboxane A2

pubblicato su: MEDICINAL CHEMISTRY - 2018

Applová Lenka, Veljović Elma, Muratović Samija, Karlíčková Jana, Macáková Kateřina, Završnik Davorka, Saso Luciano, Durić Kemal, Mladĕnka Přemysl

Insights into the phytochemistry of the cuban endemic medicinal plant phyllanthus orbicularis: fideloside, a novel bioactive 8-c-glycosyl 2,3-dihydroflavonol

pubblicato su: MOLECULES - 2019

Francioso A., Franke K., Villani C., Mosca L., D'Erme M., Frischbutter S., Brandt W., Sanchez-Lamar A., Wessjohann L.

Discovery of dihydroxyindole-2-carboxylic acid derivatives as dual allosteric HIV-1 integrase and reverse transcriptase associated ribonuclease H inhibitors

pubblicato su: ANTIVIRAL RESEARCH - 2020

Esposito F., Sechi M., Pala N., Sanna A., Koneru P. C., Kvaratskhelia M., Naesens L., Corona A., Grandi N., di Santo R., D'Amore V. M., Di Leva F. S., Novellino E., Cosconati S., Tramontano E.

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