Risultati ricerca pubblicazioni

Leveraging the cruzain S3 subsite to increase affinity for reversible covalent inhibitors

pubblicato su: BIOORGANIC CHEMISTRY - 2018

Cianni Lorenzo, Sartori Geraldo, Rosini Fabiana, De Vita Daniela, Pires Gabriel, Lopes Bianca Rebelo, Leitão Andrei, Burtoloso Antonio C B, Montanari Carlos A

Oregonin from Alnus incana bark affects DNA methyltransferases expression and mitochondrial DNA copies in mouse embryonic fibroblasts

pubblicato su: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY - 2018

Krasilnikova Jelena, Lauberte Liga, Stoyanova Elena, Abadjieva Desislava, Chervenkov Mihail, Mori Mattia, De Paolis Elisa, Mladenova Vanya, Telysheva Galina, Botta Bruno, Kistanova Elena

Synthesis and characterisation of a new benzamide-containing nitrobenzoxadiazole as a GSTP1-1 inhibitor endowed with high stability to metabolic hydrolysis

pubblicato su: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY - 2019

Di Paolo V., Fulci C., Rotili D., Sciarretta F., Lucidi A., Morozzo della Rocca B., De Luca A., Rosato A., Quintieri L., Caccuri A. M.

Efficient synthesis and first regioselective C-6 direct arylation of imidazo[2,1-c][1,2,4]triazine scaffold and their evaluation in H2O2-induced oxidative stress

pubblicato su: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 2018

Loubidi Mohammed, Jouha Jabrane, Tber Zahira, Khouili Mostafa, Suzenet Franck, Akssira Mohamed, Erdogan Mümin Alper, Köse Fadime Aydın, Dagcı Taner, Armagan Güliz, Saso Luciano, Guillaumet Gérald

9-(4'-dimethylaminophenyl)-2,6,7-trihydroxy-xanthene-3-one is a potentially novel antiplatelet drug which antagonizes the effect of thromboxane A2

pubblicato su: MEDICINAL CHEMISTRY - 2018

Applová Lenka, Veljović Elma, Muratović Samija, Karlíčková Jana, Macáková Kateřina, Završnik Davorka, Saso Luciano, Durić Kemal, Mladĕnka Přemysl

Discovery of dihydroxyindole-2-carboxylic acid derivatives as dual allosteric HIV-1 integrase and reverse transcriptase associated ribonuclease H inhibitors

pubblicato su: ANTIVIRAL RESEARCH - 2020

Esposito F., Sechi M., Pala N., Sanna A., Koneru P. C., Kvaratskhelia M., Naesens L., Corona A., Grandi N., di Santo R., D'Amore V. M., Di Leva F. S., Novellino E., Cosconati S., Tramontano E.