Daniela De Vita

Pubblicazioni

Titolo Pubblicato in Anno
On the intrinsic reactivity of highly potent trypanocidal cruzain inhibitors RSC MEDICINAL CHEMISTRY 2020
Searching for new agents active against candida albicans biofilm: a series of indole derivatives, design, synthesis and biological evaluation EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 2019
Design, synthesis, and biological evaluation of new 1-(aryl-1H-pyrrolyl)(phenyl)methyl-1H-imidazole derivatives as antiprotozoal agents JOURNAL OF MEDICINAL CHEMISTRY 2019
Comparison of different methods for the extraction of cannabinoids from cannabis NATURAL PRODUCT RESEARCH 2019
Pedicularis L. Genus. Systematics, botany, phytochemistry, chemotaxonomy, ethnopharmacology, and other PLANTS 2019
Synthesis and structure-activity relationship of nitrile-based cruzain inhibitors incorporating a trifluoroethylamine-based P2 amide replacement BIOORGANIC & MEDICINAL CHEMISTRY 2019
Towards a new application of amaranth seed oil as an agent against Candida albicans NATURAL PRODUCT RESEARCH 2019
Anti-inflammatory and antioxidant properties of dehydrated potato-derived bioactive compounds in intestinal cells INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES 2019
Tegaserod for the treatment of Irritable Bowel syndrome ANTI-INFLAMMATORY & ANTI-ALLERGY AGENTS IN MEDICINAL CHEMISTRY 2019
Design, synthesis and biochemical evaluation of novel multi-target inhibitors as potential anti-Parkinson agents EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 2018
Biological evaluation and structure-activity relationships of imidazole-based compounds as antiprotozoal agents EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 2018
Novel symmetrical benzazolyl derivatives endowed with potent anti-heparanase activity JOURNAL OF MEDICINAL CHEMISTRY 2018
Experimental study and computational modelling of cruzain cysteine protease inhibition by dipeptidyl nitriles PHYSICAL CHEMISTRY CHEMICAL PHYSICS 2018
Leveraging the cruzain S3 subsite to increase affinity for reversible covalent inhibitors BIOORGANIC CHEMISTRY 2018
Inhibition of the α-carbonic anhydrase from Vibrio cholerae with amides and sulfonamides incorporating imidazole moieties JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY 2017
New pyridine derivatives as inhibitors of acetylcholinesterase and amyloid aggregation EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 2017
A comparative study of warheads for design of cysteine protease inhibitors BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 2017
In vitro screening of 2-(1H-imidazol-1-yl)-1-phenylethanol derivatives as antiprotozoal agents and docking studies on Trypanosoma cruzi CYP51 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 2016
Discovery of in vitro antitubercular agents through in silico ligand-based approaches EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 2016
New N,N-dimethylcarbamate inhibitors of acetylcholinesterase: design synthesis and biological evaluation JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY 2016

ERC

  • LS9_8

KET

  • Life-science technologies & biotechnologies

Interessi di ricerca

  • estrazione ed analisi dei metaboliti delle piante con potenziale applicazione in ambito farmaceutico
  • estrazione di composti con applicazione farmaceutica da scarti alimentari
  • ricerca di potenziali agenti antivirali ed antiparassitari
  • ricerca di potenziali agenti antitumorali

Keywords

Piante medicinali
fitochimica
antimicrobial agents
antiviral agents
Anticancer agents
antifungal agents

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