Antonello Mai

Publications

Title Published on Year
Recent advances in epigenetic proteolysis targeting chimeras (Epi-PROTACs) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 2020
Diphenylene Iodonium Is a Noncovalent MAO Inhibitor: A Biochemical and Structural Analysis CHEMMEDCHEM 2020
HAT inhibitors in cancer therapy Histone Modifications in Therapy 2020
Lysine Acetyltransferase Inhibitors From Natural Sources FRONTIERS IN PHARMACOLOGY 2020
Identification of novel quinazoline derivatives as potent antiplasmodial agents EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 2019
Development of alkyl glycerone phosphate synthase inhibitors: Structure-activity relationship and effects on ether lipids and epithelial-mesenchymal transition in cancer cells EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 2019
Acute and chronic neurobehavioral effects of the designer drug and bath salt constituent 3,4-methylenedioxypyrovalerone in the rat JOURNAL OF PSYCHOPHARMACOLOGY 2019
Effect of α-methoxy substitution on the anti-HIV activity of dihydropyrimidin-4(3 H)-ones JOURNAL OF MEDICINAL CHEMISTRY 2019
The emerging role of epigenetics in human autoimmune disorders CLINICAL EPIGENETICS 2019
Identification of a novel quinoline-based DNA demethylating compound highly potent in cancer cells CLINICAL EPIGENETICS 2019
Sirtuins as drug targets Epigenetic Drug Discovery 2019
Epigenetic Pharmacology in Regenerative Medicine (Epi-Drugs) Epigenetics and Regeneration 2019
Amphetamine and the Smart Drug 3,4-Methylenedioxypyrovalerone (MDPV) Induce Generalization of Fear Memory in Rats FRONTIERS IN MOLECULAR NEUROSCIENCE 2019
Enzymatic and biological characterization of novel sirtuin modulators against cancer INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES 2019
Structure-reactivity relationships on substrates and inhibitors of the lysine deacylase sirtuin 2 from schistosoma mansoni (SmSirt2) JOURNAL OF MEDICINAL CHEMISTRY 2019
Epigenetic polypharmacology: a new frontier for epi-drug discovery MEDICINAL RESEARCH REVIEWS 2019
α,γ-Diketocarboxylic acids and their esters act as carbonic anhydrase IX and XII selective inhibitors ACS MEDICINAL CHEMISTRY LETTERS 2019
DNA Methylation: Biological Implications and Modulation of Its Aberrant Dysregulation The DNA, RNA, and Histone Methylomes 2019
Dissecting the role of novel EZH2 inhibitors in primary glioblastoma cell cultures: effects on proliferation, epithelial-mesenchymal transition, migration, and on the pro-inflammatory phenotype CLINICAL EPIGENETICS 2019
Inhibition of histone demethylases LSD1 and UTX regulates ERα signaling in breast cancer CANCERS 2019

ERC

  • PE5_18

KET

  • Life-science technologies & biotechnologies

Interessi di ricerca

Keywords

drug discovery
Epigenetic drugs
antiviral agents
Anticancer drugs
parasite growth inhibition

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