Risultati ricerca pubblicazioni

SMO inhibition modulates cellular plasticity and invasiveness in colorectal cancer

pubblicato su: FRONTIERS IN PHARMACOLOGY - 2018

Magistri Paolo, Battistelli Cecilia, Strippoli Raffaele, Petrucciani Niccolò, Pellinen Teijo, Rossi Lucia, Mangogna Livia, Aurello Paolo, D'Angelo Francesco, Tripodi Marco, Ramacciato Giovanni, Nigri Giuseppe

Natural products inspired modulators of cancer stem cells-specific signaling pathways notch and hedgehog

pubblicato su: CURRENT PHARMACEUTICAL DESIGN - 2018

Palermo Rocco, Ghirga Francesca, Piccioni Maria Grazia, Bernardi Flavia, Zhdanovskaya Nadezda, Infante Paola, Mori Mattia

In vivo potent BM635 analogue with improved drug-like properties

pubblicato su: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 2018

Poce Giovanna, Cocozza Martina, Alfonso Salvatore, Consalvi Sara, Venditti Giulia, Fernandez-Menendez Raquel, Bates Robert H., Barros Aguirre David, Ballell Lluis, De Logu Alessandro, Vistoli Giulio, Biava Mariangela

Naturally occurring diels-alder-type adducts from morus nigra as potent inhibitors of mycobacterium tuberculosis protein tyrosine phosphatase B

pubblicato su: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 2018

Mascarello Alessandra, Orbem Menegatti Angela Camila, Calcaterra Andrea, Martins Priscila Graziela Alves, Chiaradia-Delatorre Louise Domeneghini, D'Acquarica Ilaria, Ferrari Franco, Pau Valentina, Sanna Adriana, De Logu Alessandro, Botta Maurizio, Botta Bruno, Terenzi Hernã¡n, Mori Mattia

Oregonin from Alnus incana bark affects DNA methyltransferases expression and mitochondrial DNA copies in mouse embryonic fibroblasts

pubblicato su: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY - 2018

Krasilnikova Jelena, Lauberte Liga, Stoyanova Elena, Abadjieva Desislava, Chervenkov Mihail, Mori Mattia, De Paolis Elisa, Mladenova Vanya, Telysheva Galina, Botta Bruno, Kistanova Elena

Crystal structure of the Eg5 - K858 complex and implications for structure-based design of thiadiazole-containing inhibitors

pubblicato su: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 2018

Talapatra Sandeep K., Tham Chuin Lean, Guglielmi Paolo, Cirilli Roberto, Chandrasekaran Balakumar, Karpoormath Rajshekhar, Carradori Simone, Kozielski Frank

Lysine acetyltransferase inhibitors: structure-activity relationships and potential therapeutic implications

pubblicato su: FUTURE MEDICINAL CHEMISTRY - 2018

Fiorentino Francesco, Mai Antonello, Rotili Dante

Trends of LSD1 inhibitors in viral infections

pubblicato su: FUTURE MEDICINAL CHEMISTRY - 2018

Zwergel Clemens, Stazi Giulia, Mai Antonello, Valente Sergio

Nucleocytoplasmic export of HDAC5 and SIRT2 downregulation: two epigenetic mechanisms by which antidepressants enhance synaptic plasticity markers

pubblicato su: PSYCHOPHARMACOLOGY - 2018

Muñoz-Cobo I., Erburu M. M., Zwergel C., Cirilli R., Mai A., Valente S., Puerta E., Tordera Rosa M.

MAO inhibitors and their wider applications: a patent review

pubblicato su: EXPERT OPINION ON THERAPEUTIC PATENTS - 2018

Carradori Simone, Secci Daniela, Petzer Jacques P.

CD28 between tolerance and autoimmunity: The side effects of animal models [version 1; referees: 2 approved]

pubblicato su: F1000RESEARCH - 2018

Porciello Nicla, Kunkl Martina, Tuosto Loretta

Targeting serotonin 2A and adrenergic α1receptors for ocular antihypertensive agents. Discovery of 3,4-dihydropyrazino[1,2-b]indazol-1(2H)-one derivatives

pubblicato su: CHEMMEDCHEM - 2018

Furlotti Guido, Alisi Maria Alessandra, Cazzolla Nicola, Ceccacci Francesca, Garrone Beatrice, Gasperi Tecla, La Bella Angela, Leonelli Francesca, Loreto Maria Antonietta, Magarò Gabriele, Mangano Giorgina, Bettolo Rinaldo Marini, Masini Emanuela, Miceli Martina, Migneco Luisa Maria, Vitiello Marco

Addiction research and theory: a commentary on the surgeon general's report on alcohol, drugs, and health

pubblicato su: ADDICTION BIOLOGY - 2018

Badiani Aldo, Berridge Kent C., Heilig Markus, Nutt David J., Robinson Terry E.

Intravenous self-administration of benzydamine, a non-steroidal anti-inflammatory drug with a central cannabinoidergic mechanism of action

pubblicato su: ADDICTION BIOLOGY - 2018

Avvisati Riccardo, Meringolo Maria, Stendardo Emiliana, Malavasi Elisa, Marinelli Silvia, Badiani Aldo

The reduction in glutamate release is predictive of cognitive and emotional alterations that are corrected by the positive modulator of AMPA receptors S 47445 in perinatal stressed rats

pubblicato su: NEUROPHARMACOLOGY - 2018

Morley-Fletcher S., Zuena A. R., Mairesse J., Gatta E., Van Camp G., Bouwalerh H., Riozzi B., Battaglia G., Pittaluga A., Olivero G., Mocaer E., Bretin S., Nicoletti F., Maccari S.

Impaired repair of DNA damage is associated with autistic-like traits in rats prenatally exposed to valproic acid

pubblicato su: EUROPEAN NEUROPSYCHOPHARMACOLOGY - 2018

Servadio Michela, Manduca Antonia, Melancia Francesca, Leboffe Loris, Schiavi Sara, Campolongo Patrizia, Palmery Maura, Ascenzi Paolo, di Masi Alessandra, Trezza Viviana

Stress as risk factor for Alzheimer's disease

pubblicato su: PHARMACOLOGICAL RESEARCH - 2018

Caruso Alessandra, Nicoletti Ferdinando, Mango Dalila, Saidi Amira, Orlando Rosamaria, Scaccianoce Sergio

Collaboration between a human group and artificial intelligence can improve prediction of multiple sclerosis course. A proof-of-principle study

pubblicato su: F1000RESEARCH - 2018

Tacchella Andrea, Romano Silvia, Ferraldeschi Michela, Salvetti Marco, Zaccaria Andrea, Crisanti Andrea, Grassi Francesca

In vitro and in vivo pharmacological activities of 14-o-phenylpropyloxymorphone, a potent mixed mu/delta/kappa-opioid receptor agonist with reduced constipation in mice

pubblicato su: FRONTIERS IN PHARMACOLOGY - 2018

Lattanzi Roberta, Rief Silvia, Schmidhammer Helmut, Negri Lucia, Spetea Mariana.

Efficient synthesis and first regioselective C-6 direct arylation of imidazo[2,1-c][1,2,4]triazine scaffold and their evaluation in H2O2-induced oxidative stress

pubblicato su: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 2018

Loubidi Mohammed, Jouha Jabrane, Tber Zahira, Khouili Mostafa, Suzenet Franck, Akssira Mohamed, Erdogan Mümin Alper, Köse Fadime Aydın, Dagcı Taner, Armagan Güliz, Saso Luciano, Guillaumet Gérald

Ultramicronized palmitoylethanolamide improves learning and memory in a triple transgenic mouse model of Alzheimer's disease through a combination of anti-inflammatory and neuroprotective effects

pubblicato su: 38th Spanish Society of Pharmacology meeting/9th Spanish Society of Pharmacogenetics and Pharmacogenomics meeting. - 2018

Scuderi Caterina, Bronzuoli MARIA ROSANNA, Facchinetti Roberta, Pace Lorenzo Federico, Canese Rossella, Carpinelli Giulia, Steardo Luca, Cassano Tommaso

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