Risultati ricerca pubblicazioni

In vivo potent BM635 analogue with improved drug-like properties

pubblicato su: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 2018

Poce Giovanna, Cocozza Martina, Alfonso Salvatore, Consalvi Sara, Venditti Giulia, Fernandez-Menendez Raquel, Bates Robert H., Barros Aguirre David, Ballell Lluis, De Logu Alessandro, Vistoli Giulio, Biava Mariangela

Naturally occurring diels-alder-type adducts from morus nigra as potent inhibitors of mycobacterium tuberculosis protein tyrosine phosphatase B

pubblicato su: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 2018

Mascarello Alessandra, Orbem Menegatti Angela Camila, Calcaterra Andrea, Martins Priscila Graziela Alves, Chiaradia-Delatorre Louise Domeneghini, D'Acquarica Ilaria, Ferrari Franco, Pau Valentina, Sanna Adriana, De Logu Alessandro, Botta Maurizio, Botta Bruno, Terenzi Hernã¡n, Mori Mattia

Crystal structure of the Eg5 - K858 complex and implications for structure-based design of thiadiazole-containing inhibitors

pubblicato su: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 2018

Talapatra Sandeep K., Tham Chuin Lean, Guglielmi Paolo, Cirilli Roberto, Chandrasekaran Balakumar, Karpoormath Rajshekhar, Carradori Simone, Kozielski Frank

Novel coumarin- and quinolinone-based polycycles as cell division cycle 25-A and -C phosphatases inhibitors induce proliferation arrest and apoptosis in cancer cells

pubblicato su: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 2017

Zwergel Clemens, Czepukojc Brigitte, Evain Bana Emilie, Xu Zhanjie, Stazi Giulia, Mori Mattia, Patsilinakos Alexandros, Mai Antonello, Botta Bruno, Ragno Rino, Bagrel Denise, Kirsch Gilbert, Meiser Peter, Jacob Claus, Montenarh Mathias, Valente Sergio

From pyrrolidinyl-benzodioxane to pyrrolidinyl-pyridodioxanes, or from unselective antagonism to selective partial agonism at ?4?2 nicotinic acetylcholine receptor

pubblicato su: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 2017

Bolchi Cristiano, Bavo Francesco, Gotti Cecilia, Fumagalli Laura, Fasoli Francesca, Binda Matteo, Mucchietto Vanessa, Sciaccaluga Miriam, Plutino Simona, Fucile Sergio, Pallavicini Marco

Efficient synthesis and first regioselective C-6 direct arylation of imidazo[2,1-c][1,2,4]triazine scaffold and their evaluation in H2O2-induced oxidative stress

pubblicato su: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 2018

Loubidi Mohammed, Jouha Jabrane, Tber Zahira, Khouili Mostafa, Suzenet Franck, Akssira Mohamed, Erdogan Mümin Alper, Köse Fadime Aydın, Dagcı Taner, Armagan Güliz, Saso Luciano, Guillaumet Gérald

Evaluation of the cellular protection by novel spiropyrazole compounds in dopaminergic cell death

pubblicato su: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 2021

Zaiter Jamila, Hibot Achraf, Hafid Abderrafia, Khouili Mostafa, Neves Claudia M. B., Simões Mário M. Q., Neves M. Graça P. M. S., Faustino M. Amparo F., Dagci Taner, Saso Luciano, Armagan Güliz