Francesco Fiorentino | Ricerc@Sapienza

Pubblicazioni

Titolo	Pubblicato in	Anno
Transcriptomic and genomic studies classify NKL54 as a histone deacetylase inhibitor with indirect influence on MEF2-dependent transcription	NUCLEIC ACIDS RESEARCH	2022
Novel non-covalent LSD1 inhibitors endowed with anticancer effects in leukemia and solid tumor cellular models	EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY	2022
Sirtuin modulators: past, present, and future perspectives	FUTURE MEDICINAL CHEMISTRY	2022
Therapeutic Potential and Activity Modulation of the Protein Lysine Deacylase Sirtuin 5	JOURNAL OF MEDICINAL CHEMISTRY	2022
Mass Spectrometry Analysis of Dynamics and Interactions of the LPS Translocon LptDE	Lipopolysaccharide Transport	2022
Modulation of virulence-associated traits in Aspergillus fumigatus by BET Inhibitor JQ1	MICROORGANISMS	2022
The two-faced role of sirt6 in cancer	CANCERS	2021
Anti-influenza A virus activity and structure–activity relationship of a series of nitrobenzoxadiazole derivatives	JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY	2021
Mass spectrometry enables the discovery of inhibitors of an LPS transport assembly via disruption of protein-protein interactions	CHEMICAL COMMUNICATIONS	2021
NaViA: A Program for the Visual Analysis of Complex Mass Spectra	BIOINFORMATICS	2021
Dynamics of an LPS translocon induced by substrate and an antimicrobial peptide	NATURE CHEMICAL BIOLOGY	2021
Anionic Dendritic Polyglycerol for Protein Purification and Delipidation	ACS APPLIED POLYMER MATERIALS	2021
Mass spectrometry informs the structure and dynamics of membrane proteins involved in lipid and drug transport	CURRENT OPINION IN STRUCTURAL BIOLOGY	2021
Emerging Therapeutic Potential of SIRT6 Modulators	JOURNAL OF MEDICINAL CHEMISTRY	2021
Assembly and regulation of the chlorhexidine-specific efflux pump AceI	PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA	2020
Structural Basis of Tail-Anchored Membrane Protein Biogenesis by the GET Insertase Complex	MOLECULAR CELL	2020
Investigating the Conformational Dynamics of the Outer Membrane LPS Translocon LptDE	BIOPHYSICAL JOURNAL	2020
HAT inhibitors in cancer therapy	Histone Modifications in Therapy	2020
Lysine Acetyltransferase Inhibitors From Natural Sources	FRONTIERS IN PHARMACOLOGY	2020
The Different Effects of Substrates and Nucleotides on the Complex Formation of ABC Transporters	STRUCTURE	2019

ERC

LS1_1
LS1_13
PE5_18

Keywords

medicinal chemistry

biophysical chemistry

epigenetics

antimicrobial resistance

high resolution mass spectrometry