| Titolo |
Pubblicato in |
Anno |
| First-in-Class Selenium-Containing Potent Serotonin Receptor 5-HT6 Agents with a Beneficial Neuroprotective Profile against Alzheimer's Disease |
JOURNAL OF MEDICINAL CHEMISTRY |
2024 |
| Theileria parasites sequester host eIF5A to escape elimination by host-mediated autophagy |
NATURE COMMUNICATIONS |
2024 |
| Uracil- and Pyridine-Containing HDAC Inhibitors Displayed Cytotoxicity in Colorectal and Glioblastoma Cancer Stem Cells |
CHEMMEDCHEM |
2024 |
| Selenium-containing compounds: a new hope for innovative treatments in Alzheimer’s disease and Parkinson’s disease |
DRUG DISCOVERY TODAY |
2024 |
| Pharmacological Activation of SIRT3 Modulates the Response of Cancer Cells to Acidic pH |
PHARMACEUTICALS |
2024 |
| Pyrimidine thioethers: A novel class of antidepressant agents, endowed with anxiolytic, performance enhancing and nootropic activity |
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY |
2023 |
| LSD1 inhibitors for cancer treatment: Focus on multi-target agents and compounds in clinical trials |
FRONTIERS IN PHARMACOLOGY |
2023 |
| GreenMedChem- the challenge in the next decade toward eco-friendly compounds and processes in drug design |
GREEN CHEMISTRY |
2023 |
| Novel 1,4-Dihydropyridines as Specific Binders and Activators of SIRT3 Impair Cell Viability and Clonogenicity and Downregulate Hypoxia-Induced Targets in Cancer Cells |
JOURNAL OF MEDICINAL CHEMISTRY |
2023 |
| Histone deacetylase 10: A polyamine deacetylase from the crystal structure to the first inhibitors |
CURRENT OPINION IN STRUCTURAL BIOLOGY |
2023 |
| Molecular Docking Assessment of Cathinones as 5-HT2AR Ligands: Developing of Predictive Structure-Based Bioactive Conformations and Three-Dimensional Structure-Activity Relationships Models for Future Recognition of Abuse Drugs |
MOLECULES |
2023 |
| Essential Oils from Mediterranean Plants Inhibit In Vitro Monocyte Adhesion to Endothelial Cells from Umbilical Cords of Females with Gestational Diabetes Mellitus |
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES |
2023 |
| Heterocycle-containing tranylcypromine derivatives endowed with high anti-LSD1 activity |
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY |
2022 |
| Current HDAC Inhibitors in Clinical Trials |
CHIMIA |
2022 |
| Effects of Structurally Different HDAC Inhibitors against Trypanosoma cruzi, Leishmania, and Schistosoma mansoni |
ACS INFECTIOUS DISEASES |
2022 |
| Bovine serum amine oxidase and polyamine analogues: chemical synthesis and biological evaluation integrated with molecular docking and 3-D QSAR studies |
JOURNAL OF CHEMICAL INFORMATION AND MODELING |
2022 |
| Seleno-vs. thioether triazine derivatives in search for new anticancer agents overcoming multidrug resistance in lymphoma |
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY |
2022 |
| Potent and Specific Activators for Mitochondrial Sirtuins Sirt3 and Sirt5 |
JOURNAL OF MEDICINAL CHEMISTRY |
2022 |
| Chemically Diverse S. mansoni HDAC8 Inhibitors Reduced Viability in Worm Larval and Adult Stages |
CHEMMEDCHEM |
2022 |
| PD-L1 small-molecule modulators: a new hope in epigenetic-based multidrug cancer therapy? |
DRUG DISCOVERY TODAY |
2022 |
