Rossella Fioravanti | Ricerc@Sapienza

Pubblicazioni

Titolo	Pubblicato in	Anno
First-in-Class Selenium-Containing Potent Serotonin Receptor 5-HT6 Agents with a Beneficial Neuroprotective Profile against Alzheimer's Disease	JOURNAL OF MEDICINAL CHEMISTRY	2024
Theileria parasites sequester host eIF5A to escape elimination by host-mediated autophagy	NATURE COMMUNICATIONS	2024
Pyrimidine thioethers: A novel class of antidepressant agents, endowed with anxiolytic, performance enhancing and nootropic activity	EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY	2023
LSD1 inhibitors for cancer treatment: Focus on multi-target agents and compounds in clinical trials	FRONTIERS IN PHARMACOLOGY	2023
GreenMedChem- the challenge in the next decade toward eco-friendly compounds and processes in drug design	GREEN CHEMISTRY	2023
Novel 1,4-Dihydropyridines as Specific Binders and Activators of SIRT3 Impair Cell Viability and Clonogenicity and Downregulate Hypoxia-Induced Targets in Cancer Cells	JOURNAL OF MEDICINAL CHEMISTRY	2023
Histone deacetylase 10: A polyamine deacetylase from the crystal structure to the first inhibitors	CURRENT OPINION IN STRUCTURAL BIOLOGY	2023
Molecular Docking Assessment of Cathinones as 5-HT2AR Ligands: Developing of Predictive Structure-Based Bioactive Conformations and Three-Dimensional Structure-Activity Relationships Models for Future Recognition of Abuse Drugs	MOLECULES	2023
Essential Oils from Mediterranean Plants Inhibit In Vitro Monocyte Adhesion to Endothelial Cells from Umbilical Cords of Females with Gestational Diabetes Mellitus	INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES	2023
Heterocycle-containing tranylcypromine derivatives endowed with high anti-LSD1 activity	JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY	2022
Current HDAC Inhibitors in Clinical Trials	CHIMIA	2022
Effects of Structurally Different HDAC Inhibitors against Trypanosoma cruzi, Leishmania, and Schistosoma mansoni	ACS INFECTIOUS DISEASES	2022
Bovine serum amine oxidase and polyamine analogues: chemical synthesis and biological evaluation integrated with molecular docking and 3-D QSAR studies	JOURNAL OF CHEMICAL INFORMATION AND MODELING	2022
Seleno-vs. thioether triazine derivatives in search for new anticancer agents overcoming multidrug resistance in lymphoma	EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY	2022
Potent and Specific Activators for Mitochondrial Sirtuins Sirt3 and Sirt5	JOURNAL OF MEDICINAL CHEMISTRY	2022
Chemically Diverse S. mansoni HDAC8 Inhibitors Reduced Viability in Worm Larval and Adult Stages	CHEMMEDCHEM	2022
PD-L1 small-molecule modulators: a new hope in epigenetic-based multidrug cancer therapy?	DRUG DISCOVERY TODAY	2022
Novel pyridine-containing histone deacetylase inhibitors strongly arrest proliferation, induce apoptosis and modulate miRNAs in cancer cells	EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY	2022
Selenium-Containing Agents Acting on Cancer—A New Hope?	PHARMACEUTICS	2022
Novel quinoline compounds active in cancer cells through coupled DNA methyltransferase inhibition and degradation	CANCERS	2020

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Life-science technologies & biotechnologies

Laboratori di ricerca

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