Mariangela Biava

Pubblicazioni

Titolo Pubblicato in Anno
Development of MmpL3 inhibitors for tuberculosis treatment Medicinal Chemistry approaches to tuberculosis and trypanosomiasis 2019
In vivo potent BM635 analogue with improved drug-like properties EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 2018
Introduction to COX inhibitors FUTURE MEDICINAL CHEMISTRY 2018
In vitro comprehensive analysis of VA692 a new chemical entity for the treatment of osteoarthritis INTERNATIONAL IMMUNOPHARMACOLOGY 2018
1,5-Diarylpyrroles as potent antitubercular and anti-inflammatory agents CHEMISTRY OF HETEROCYCLIC COMPOUNDS 2017
Pharmaceutical salt of BM635 with improved bioavailability EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES 2017
Synthesis and biological evaluation of fluorinated 1,5-diarylpyrrole-3-alkoxyethyl ether derivatives as selective COX-2 inhibitors endowed with anti-inflammatory activity EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 2016
(E)-3-Heteroarylidenechroman-4-ones as potent and selective monoamine oxidase-B inhibitors EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 2016
A series of COX-2 inhibitors endowed with NO-releasing properties: synthesis, biological evaluation, and docking analysis CHEMMEDCHEM 2016
MmpL3 inhibitors: diverse chemical scaffolds inhibit the same target MINI-REVIEWS IN MEDICINAL CHEMISTRY 2016
A novel antimycobacterial compound acts as an intracellular iron chelator ANTIMICROBIAL AGENTS AND CHEMOTHERAPY 2015
Activity of lipophilic and hydrophilic drugs against dormant and replicating mycobacterium tuberculosis JOURNAL OF ANTIBIOTICS 2015
N-((1,3-diphenyl-1H-pyrazol-4-yl)methyl)anilines: a novel class of anti-RSV agents BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 2015
COX inhibitors: a patent review (2011 - 2014) EXPERT OPINION ON THERAPEUTIC PATENTS 2015
Chondroprotective effect of three different classes of anti-inflammatory agents on human osteoarthritic chondrocytes exposed to IL-1β INTERNATIONAL IMMUNOPHARMACOLOGY 2015
Overcoming drug resistance for tuberculosis FUTURE MICROBIOLOGY 2015
Synthesis, biological evaluation and docking analysis of a new series of methylsulfonyl and sulfamoyl acetamides and ethyl acetates as potent COX-2 inhibitors BIOORGANIC & MEDICINAL CHEMISTRY 2015
Synthesis, biological evaluation and docking analysis of a new series of methylsulfonyl and sulfamoyl acetamides and ethyl acetates as potent COX-2 inhibitors BIOORGANIC & MEDICINAL CHEMISTRY 2015

Progetti di Ricerca

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