Arianna Granese | Ricerc@Sapienza

Pubblicazioni

Titolo	Pubblicato in	Anno
Development of N-(4-(1 H-Imidazol-1-yl)phenyl)-4-chlorobenzenesulfonamide, a Novel Potent Inhibitor of β-Catenin with Enhanced Antitumor Activity and Metabolic Stability	JOURNAL OF MEDICINAL CHEMISTRY	2024
Novel therapeutic opportunities for Toxoplasma gondii, Trichomonas vaginalis, and Giardia intestinalis infections	EXPERT OPINION ON THERAPEUTIC PATENTS	2023
Synthesis and Evaluation of Thymol-Based Synthetic Derivatives as Dual-Action Inhibitors against Different Strains of H. pylori and AGS Cell Line	MOLECULES	2021
A novel class of dual-acting DCH-CORMs counteracts oxidative stress-induced inflammation in human primary tenocytes	ANTIOXIDANTS	2021
Phytochemical analyses and pharmacological screening of Neem oil	SOUTH AFRICAN JOURNAL OF BOTANY	2019
Analytical procedures for secondary metabolites determination: recent trends and future perspectives	LETTERS IN DRUG DESIGN & DISCOVERY	2018
Antimicrobial activity, synergism and inhibition of germ tube formation by Crocus sativus-derived compounds against Candida spp	JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY	2016
(Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies	JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY	2015
Bioactive compounds of Crocus sativus L. and their semisynthetic derivatives as promising anti-Helicobacter pylori, anti-malarial and anti-leishmanial agents	JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY	2015
Nitric oxide donors and selective carbonic anhydrase inhibitors: A dual pharmacological approach for the treatment of glaucoma, cancer and osteoporosis	MOLECULES	2015

ERC

LS1
LS7_4
PE4_2
PE4_5
PE5

KET

Life-science technologies & biotechnologies

Interessi di ricerca

Sintesi di composti come inibori selettivi delle monoamminossidasi, MAO-A e MAO-B.

Sintesi di composti attivi sull'Helicobacter pylori, su ceppi di Candida e su Toxoplasma.

Sintesi di composti come inibitori/modulatori delle istone acetiltransferasi (HAT)

Keywords

anticancer agent

neuroprotective agents

drug design and discovery