Dante Rotili

Pubblicazioni

Titolo Pubblicato in Anno
Effect of α-methoxy substitution on the anti-HIV activity of dihydropyrimidin-4(3 H)-ones JOURNAL OF MEDICINAL CHEMISTRY 2019
Sirtuins as drug targets Epigenetic Drug Discovery 2019
Gold nanoparticles and nanorods in nuclear medicine: a mini review APPLIED SCIENCES 2019
Enzymatic and biological characterization of novel sirtuin modulators against cancer INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES 2019
Structure-reactivity relationships on substrates and inhibitors of the lysine deacylase sirtuin 2 from schistosoma mansoni (SmSirt2) JOURNAL OF MEDICINAL CHEMISTRY 2019
Epigenetic polypharmacology: a new frontier for epi-drug discovery MEDICINAL RESEARCH REVIEWS 2019
α,γ-Diketocarboxylic acids and their esters act as carbonic anhydrase IX and XII selective inhibitors ACS MEDICINAL CHEMISTRY LETTERS 2019
DNA Methylation: Biological Implications and Modulation of Its Aberrant Dysregulation The DNA, RNA, and Histone Methylomes 2019
Inhibition of histone demethylases LSD1 and UTX regulates ERα signaling in breast cancer CANCERS 2019
Histone deacetylase inhibitors exert anti-tumor effects on human adherent and stem-like glioma cells 11 Medical and Health Sciences 1112 Oncology and Carcinogenesis CLINICAL EPIGENETICS 2019
Comparison of the effects of synthetic and plant-derived mTOR regulators on healthy human ovarian cells EUROPEAN JOURNAL OF PHARMACOLOGY 2019
Effects of glutathione transferase-targeting nitrobenzoxadiazole compounds in relation to PD-L1 status in human melanoma cells CHEMOTHERAPY 2019
H19-dependent transcriptional regulation of β3 and β4 integrins upon estrogen and hypoxia favors metastatic potential in prostate cancer INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES 2019
Synthesis and characterisation of a new benzamide-containing nitrobenzoxadiazole as a GSTP1-1 inhibitor endowed with high stability to metabolic hydrolysis JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY 2019
Histone Acetyltransferase Enzymes: From Biological Implications to Most Relevant Inhibitors Topics in Medicinal Chemistry 2019
Disruptor of telomeric silencing 1-like (DOT1L): disclosing a new class of non-nucleoside inhibitors by means of ligand-based and structure-based approaches JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN 2018
RIP1-HAT1-SirT complex identification and targeting in treatment and prevention of cancer CLINICAL CANCER RESEARCH 2018
Mass spectrometry characterization of DOTA-Nimotuzumab conjugate as precursor of an innovative β − tracer suitable in radio-guided surgery JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS 2018
KAT3B-p300 and H3AcK18/H3AcK14 levels are prognostic markers for kidney ccRCC tumor aggressiveness and target of KAT inhibitor CPTH2 CLINICAL EPIGENETICS 2018
Lysine acetyltransferase inhibitors: structure-activity relationships and potential therapeutic implications FUTURE MEDICINAL CHEMISTRY 2018

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