| Titolo |
Pubblicato in |
Anno |
| Pyrimidine thioethers: A novel class of antidepressant agents, endowed with anxiolytic, performance enhancing and nootropic activity |
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY |
2023 |
| Systematic Design of Adenosine Analogs as Inhibitors of a Clostridioides difficile-Specific DNA Adenine Methyltransferase Required for Normal Sporulation and Persistence |
JOURNAL OF MEDICINAL CHEMISTRY |
2023 |
| METTL3 from Target Validation to the First Small-Molecule Inhibitors: A Medicinal Chemistry Journey |
JOURNAL OF MEDICINAL CHEMISTRY |
2023 |
| Simultaneous administration of EZH2 and BET inhibitors inhibits proliferation and clonogenic ability of metastatic prostate cancer cells |
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY |
2023 |
| GreenMedChem- the challenge in the next decade toward eco-friendly compounds and processes in drug design |
GREEN CHEMISTRY |
2023 |
| Role of SIRT3 in Microgravity Response: A New Player in Muscle Tissue Recovery |
CELLS |
2023 |
| Antihistamines, phenothiazine-based antipsychotics, and tricyclic antidepressants potently activate pharmacologically relevant human carbonic anhydrase isoforms II and VII |
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY |
2023 |
| Emerging Roles of SIRT5 in Metabolism, Cancer, and SARS-CoV-2 Infection |
CELLS |
2023 |
| Native mass spectrometry-directed drug discovery: Recent advances in investigating protein function and modulation |
DRUG DISCOVERY TODAY |
2023 |
| Hydrophilic gold nanoparticles as Anti-PD-L1 antibody carriers. Synthesis and interface properties |
PARTICLE & PARTICLE SYSTEMS CHARACTERIZATION |
2022 |
| Multimodal evaluation of 19F-BPA internalization in pancreatic cancer cells for boron capture and proton therapy potential applications |
PHYSICA MEDICA |
2022 |
| Biochemical functions and clinical characterizations of the sirtuins in diabetes-induced retinal pathologies |
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES |
2022 |
| Transcriptomic and genomic studies classify NKL54 as a histone deacetylase inhibitor with indirect influence on MEF2-dependent transcription |
NUCLEIC ACIDS RESEARCH |
2022 |
| The Nitrobenzoxadiazole Derivative NBDHEX Behaves as Plasmodium falciparum Gametocyte Selective Inhibitor with Malaria Parasite Transmission Blocking Activity |
PHARMACEUTICALS |
2022 |
| A potent HDAC inhibitor blocks Toxoplasma gondii tachyzoite growth and profoundly disrupts parasite gene expression |
INTERNATIONAL JOURNAL OF ANTIMICROBIAL AGENTS |
2022 |
| Neuroprotective effects of PARP inhibitors in Drosophila models of Alzheimer’s disease |
CELLS |
2022 |
| Novel non-covalent LSD1 inhibitors endowed with anticancer effects in leukemia and solid tumor cellular models |
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY |
2022 |
| Sirtuin modulators: past, present, and future perspectives |
FUTURE MEDICINAL CHEMISTRY |
2022 |
| Effects of Structurally Different HDAC Inhibitors against Trypanosoma cruzi, Leishmania, and Schistosoma mansoni |
ACS INFECTIOUS DISEASES |
2022 |
| Therapeutic Potential and Activity Modulation of the Protein Lysine Deacylase Sirtuin 5 |
JOURNAL OF MEDICINAL CHEMISTRY |
2022 |
