Giancarlo Fabrizi

Pubblicazioni

Titolo Pubblicato in Anno
Synthesis of functionalised 2,3-dihydroquinolin-4(1H)-ones vs. quinoline or N-alkenylindole derivatives through sequential reactions of 2-alkynylanilines with ketones ORGANIC & BIOMOLECULAR CHEMISTRY 2021
Phytocomplex characterization and biological evaluation of powdered fruits and leaves from Elaeagnus angustifolia MOLECULES 2020
Identification of novel quinazoline derivatives as potent antiplasmodial agents EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 2019
Development of alkyl glycerone phosphate synthase inhibitors: Structure-activity relationship and effects on ether lipids and epithelial-mesenchymal transition in cancer cells EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 2019
Chalcones and chalcone-mimetic derivatives as Notch inhibitors in a model of T-cell Acute Lymphoblastic Leukemia ACS MEDICINAL CHEMISTRY LETTERS 2019
Stereo- and regioselective gold(i)-catalyzed hydroamination of 2-(arylethynyl)pyridines with anilines ORGANIC & BIOMOLECULAR CHEMISTRY 2019
Palladium-catalyzed C12-selective direct arylation of [1,2-c] quinazolin-6(5H)-ones SYNTHESIS 2019
Synthesis of pyrano[2,3-: F] chromen-2-ones vs. pyrano[3,2-g] chromen-2-ones through site controlled gold-catalyzed annulations ORGANIC & BIOMOLECULAR CHEMISTRY 2019
Palladium-Catalyzed Cascade Approach to 12-(Aryl)indolo[1,2- c ]quin­azolin-6(5 H )-ones SYNTHESIS 2018
Copper-catalyzed C-N bond formation via C-H functionalization: facile synthesis of multisubstituted imidazo[1,2- a ]pyridines from N -(2-pyridinyl)enaminones SYNTHESIS 2018
Synthesis of indolo[1,2-c]quinazolines from 2-alkynylaniline derivatives through Pd-catalyzed indole formation/cyclization with N,N-dimethylformamide dimethyl acetal BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY 2018
Design, palladium-catalyzed synthesis, and biological investigation of 2-substituted 3-aroylquinolin-4(1H)-ones as inhibitors of the Hedgehog signaling pathway. JOURNAL OF MEDICINAL CHEMISTRY 2017
2-(Aminomethyl)-3-arylindoles from 3-(o-Trifluoroacetamidoaryl)-1-propargylic Alcohols, Aryl Halides, and Amines: A Domino Palladium-Catalyzed Three-Component Approach SYNTHESIS 2017
Construction of the 1,5-benzodiazepine skeleton from o-phenylendiamine and propargylic alcohols via a domino gold-catalyzed hydroamination/cyclization process ORGANIC LETTERS 2016
Total Synthesis of (±)-Kuwanol E JOURNAL OF NATURAL PRODUCTS 2016
A facile palladium-catalyzed route to 2,5,7-trisubstituted indoles TETRAHEDRON 2015
Pd- and Rh-catalyzed hydroarylation of γ-(2-methoxycarbonylphenyl)propargylic alcohols: approaches to 4- or 5-substituted seven-membered benzolactones and 3,3-disubstituted phthalides JOURNAL OF ORGANIC CHEMISTRY 2015
Palladium-catalyzed nucleophilic substitution of propargylic carbonates and meldrum's acid derivatives EUROPEAN JOURNAL OF ORGANIC CHEMISTRY 2015
Synthesis of free NH 2-(aminomethyl)indoles through copper-catalyzed reaction of 3-(ortho-trifluoroacetamidophenyl)-1-propargylic alcohols with amines and palladium/copper- cocatalyzed domino three-component Sonogashira cross-coupling/cyclization/substitution reactions ADVANCED SYNTHESIS & CATALYSIS 2015

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