Giancarlo Fabrizi

Pubblicazioni

Titolo Pubblicato in Anno
Development of alkyl glycerone phosphate synthase inhibitors: Structure-activity relationship and effects on ether lipids and epithelial-mesenchymal transition in cancer cells EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 2019
Chalcones and chalcone-mimetic derivatives as Notch inhibitors in a model of T-cell Acute Lymphoblastic Leukemia ACS MEDICINAL CHEMISTRY LETTERS 2019
Stereo- and regioselective gold(i)-catalyzed hydroamination of 2-(arylethynyl)pyridines with anilines ORGANIC & BIOMOLECULAR CHEMISTRY 2019
Palladium-catalyzed C12-selective direct arylation of [1,2-c] quinazolin-6(5H)-ones SYNTHESIS 2019
Synthesis of pyrano[2,3-: F] chromen-2-ones vs. pyrano[3,2-g] chromen-2-ones through site controlled gold-catalyzed annulations ORGANIC & BIOMOLECULAR CHEMISTRY 2019
Palladium-Catalyzed Cascade Approach to 12-(Aryl)indolo[1,2- c ]quin­azolin-6(5 H )-ones SYNTHESIS 2018
Copper-catalyzed C-N bond formation via C-H functionalization: facile synthesis of multisubstituted imidazo[1,2- a ]pyridines from N -(2-pyridinyl)enaminones SYNTHESIS 2018
Synthesis of indolo[1,2-c]quinazolines from 2-alkynylaniline derivatives through Pd-catalyzed indole formation/cyclization with N,N-dimethylformamide dimethyl acetal BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY 2018
Design, palladium-catalyzed synthesis, and biological investigation of 2-substituted 3-aroylquinolin-4(1H)-ones as inhibitors of the Hedgehog signaling pathway. JOURNAL OF MEDICINAL CHEMISTRY 2017
2-(Aminomethyl)-3-arylindoles from 3-(o-Trifluoroacetamidoaryl)-1-propargylic Alcohols, Aryl Halides, and Amines: A Domino Palladium-Catalyzed Three-Component Approach SYNTHESIS 2017
Construction of the 1,5-benzodiazepine skeleton from o-phenylendiamine and propargylic alcohols via a domino gold-catalyzed hydroamination/cyclization process ORGANIC LETTERS 2016
Total Synthesis of (±)-Kuwanol E JOURNAL OF NATURAL PRODUCTS 2016
A facile palladium-catalyzed route to 2,5,7-trisubstituted indoles TETRAHEDRON 2015
Pd- and Rh-catalyzed hydroarylation of γ-(2-methoxycarbonylphenyl)propargylic alcohols: approaches to 4- or 5-substituted seven-membered benzolactones and 3,3-disubstituted phthalides JOURNAL OF ORGANIC CHEMISTRY 2015
Palladium-catalyzed nucleophilic substitution of propargylic carbonates and meldrum's acid derivatives EUROPEAN JOURNAL OF ORGANIC CHEMISTRY 2015
Synthesis of free NH 2-(aminomethyl)indoles through copper-catalyzed reaction of 3-(ortho-trifluoroacetamidophenyl)-1-propargylic alcohols with amines and palladium/copper- cocatalyzed domino three-component Sonogashira cross-coupling/cyclization/substitution reactions ADVANCED SYNTHESIS & CATALYSIS 2015

© Università degli Studi di Roma "La Sapienza" - Piazzale Aldo Moro 5, 00185 Roma