Risultati ricerca pubblicazioni

In-vitro evaluation of different antimicrobial combinations with and without colistin against carbapenem-resistant acinetobacter baumannii

pubblicato su: MOLECULES - 2019

Oliva Alessandra, Garzoli Stefania, De Angelis Massimiliano, Marzuillo Carolina, Vullo Vincenzo, Mastroianni Claudio M., Ragno Rino

Machine learning analyses on data including essential oil chemical composition and in vitro experimental antibiofilm activities against Staphylococcus species.

pubblicato su: MOLECULES - 2019

Patsilinakos A, Artini M, Papa R, Sabatino M, Božović M, Garzoli S, Vrenna G, Buzzi R, Manfredini S, Selan L, Ragno R

Chemical investigations of male and female leaf extracts from Schinus molle L

pubblicato su: NATURAL PRODUCT RESEARCH - 2019

Garzoli Stefania, Laghezza Masci Valentina, Turchetti Giovanni, Pesci Lorenzo, Tiezzi Antonio, Ovidi Elisa

Chemical composition and antimicrobial activity of essential oil of Helichrysum italicum (Roth) G. Don fil. (Asteraceae) from Montenegro

pubblicato su: NATURAL PRODUCT RESEARCH - 2019

Oliva A., Garzoli S., Sabatino M., Tadic V., Costantini S., Ragno R., Bozovic M.

Chemical investigation of a biologically active schinus molle L. leaf extract

pubblicato su: JOURNAL OF ANALYTICAL METHODS IN CHEMISTRY - 2019

Garzoli S., Masci V. L., Ovidi E., Turchetti G., Zago D., Tiezzi A.

Liquid and vapour phase of lavandin (Lavandula × intermedia) essential oil: chemical composition and antimicrobial activity

pubblicato su: MOLECULES - 2019

Garzoli S., Turchetti G., Giacomello P., Tiezzi A., Masci V. L., Ovidi E.

Ab-initio and experimental study of pentose sugar dehydration mechanism in the gas phase

pubblicato su: CARBOHYDRATE RESEARCH - 2018

Antonini L., Garzoli S., Ricci A., Troiani A., Salvitti C., Giacomello P., Ragno R., Patsilinakos Alexandros, Di Rienzo B., Pepi F.

Antimicrobial and antibiofilm activity and machine learning classification analysis of essential oils from different mediterranean plants against pseudomonas aeruginosa

pubblicato su: MOLECULES - 2018

Artini Marco, Patsilinakos Alexandros, Papa Rosanna, Božović Mijat, Sabatino Manuela, Garzoli Stefania, Vrenna Gianluca, Tilotta Marco, Pepi Federico, Ragno Rino, Selan Laura

From ascorbic acid to furan derivatives: the gas phase acid catalyzed degradation of vitamin C

pubblicato su: PHYSICAL CHEMISTRY CHEMICAL PHYSICS - 2018

Cimino Paola, Troiani Anna, Pepi Federico, Garzoli Stefania, Salvitti Chiara, Di Rienzo Brunella, Barone Vincenzo, Ricci Andreina

High potency of melaleuca alternifolia essential oil against multi-drug resistant gram-negative bacteria and methicillin-resistant staphylococcus aureus

pubblicato su: MOLECULES - 2018

Oliva Alessandra, Costantini Silvia, De Angelis Massimiliano, Garzoli Stefania, Božović Mijat, Mascellino Maria Teresa, Vullo Vincenzo, Ragno Rino

Analytical procedures for secondary metabolites determination: recent trends and future perspectives

pubblicato su: LETTERS IN DRUG DESIGN & DISCOVERY - 2018

Menghini Luigi, Bellagamba Giuseppe, Marcelli Fabiana, Armellani Luca, Granese Arianna, DE LUCA Elisa, Cifelli Roberta, Nilgun Zengin Kucukercan, Abdurrahman Aktumsek, Gokhan Zengin

High-performance liquid chromatography enantioseparation of chiral 2-(benzylsulfinyl)benzamide derivatives on cellulose tris(3,5-dichlorophenylcarbamate) chiral stationary phase

pubblicato su: JOURNAL OF CHROMATOGRAPHY A - 2020

Carradori S., Secci D., Guglielmi P., Pierini M., Cirilli R.

1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors

pubblicato su: JOURNAL OF MEDICINAL CHEMISTRY - 2020

D'Ascenzio M., Secci D., Carradori S., Zara S., Guglielmi P., Cirilli R., Pierini M., Poli G., Tuccinardi T., Angeli A., Supuran C. T.

Chalcones: Unearthing their therapeutic possibility as monoamine oxidase B inhibitors

pubblicato su: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 2020

Guglielmi Paolo, Mathew Bijo, Secci Daniela, Carradori Simone

Antimalarial Agents from Medicinal Plant and Fungal Sources

pubblicato su: Plant-derived Bioactives. Production, Properties and Therapeutic Applications - 2020

Luisi Grazia, Carradori Simone, Grande Rossella, Secci Daniela, Guglielmi Paolo

Synthesis and evaluation of a large library of nitroxoline derivatives as pancreatic cancer antiproliferative agents

pubblicato su: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY - 2020

Veschi Serena, Carradori Simone, De Lellis Laura, Florio Rosalba, Brocco Davide, Secci Daniela, Guglielmi Paolo, Spano Mattia, Sobolev Anatoly P., Cama Alessandro

Novel therapies for glaucoma: a patent review (2013-2019)

pubblicato su: EXPERT OPINION ON THERAPEUTIC PATENTS - 2019

Guglielmi Paolo, Carradori Simone, Campestre Cristina, Poce Giovanna

The up-regulation of oxidative stress as a potential mechanism of novel MAO-B inhibitors for glioblastoma treatment

pubblicato su: MOLECULES - 2019

Marconi G. D., Gallorini M., Carradori S., Guglielmi P., Cataldi A., Zara S.

Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold

pubblicato su: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY - 2019

Rotondi G., Guglielmi P., Carradori S., Secci D., De Monte C., De Filippis B., Maccallini C., Amoroso R., Cirilli R., Akdemir A., Angeli A., Supuran C. T.

Novel approaches to the discovery of selective human monoamine oxidase-B inhibitors: is there room for improvement?

pubblicato su: EXPERT OPINION ON DRUG DISCOVERY - 2019

Guglielmi P., Carradori S., Ammazzalorso A., Secci D.

Kinesin Eg5 targeting inhibitors as a new strategy for gastric adenocarcinoma treatment

pubblicato su: MOLECULES - 2019

Marconi G. D., Carradori S., Ricci A., Guglielmi P., Cataldi A., Zara S.

Mechanisms of action of carbonic anhydrase inhibitors: compounds that bind “out of the binding site” and compounds with an unknown mechanism of action

pubblicato su: Carbonic Anhydrases Biochemistry and Pharmacology of an Evergreen Pharmaceutical Target - 2019

Carradori Simone, Guglielmi Paolo

Magnetic metal−organic framework composite by fast and facile mechanochemical process

pubblicato su: INORGANIC CHEMISTRY - 2018

Bellusci M., Guglielmi P., Masi Andrea, Padella F., Singh G., Yaacoub N., Peddis D., Secci D.

Crystal structure of the Eg5 - K858 complex and implications for structure-based design of thiadiazole-containing inhibitors

pubblicato su: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 2018

Talapatra Sandeep K., Tham Chuin Lean, Guglielmi Paolo, Cirilli Roberto, Chandrasekaran Balakumar, Karpoormath Rajshekhar, Carradori Simone, Kozielski Frank

Food and COVID-19: preventive/co-therapeutic strategies explored by current clinical trials and in silico studies

pubblicato su: FOODS - 2020

Di Matteo Giacomo, Spano Mattia, Grosso Michela, Salvo Andrea, Ingallina Cinzia, Russo Mariateresa, Ritieni Alberto, Mannina Luisa

Characterization of local products for their industrial use: the case of italian potato cultivars analyzed by untargeted and targeted methodologies

pubblicato su: FOODS - 2020

Ingallina Cinzia, Spano Mattia, Sobolev Anatoly P, Esposito Cristina, Santarcangelo Cristina, Baldi Alessandra, Daglia Maria, Mannina Luisa

Extra-virgin olive oils from nine italian regions: an ¹H NMR-chemometric characterization

pubblicato su: METABOLITES - 2019

Ingallina Cinzia, Cerreto Antonella, Mannina Luisa, Circi Simone, Vista Silvia, Capitani Donatella, Spano Mattia, Sobolev Anatoly P, Marini Federico

Use of NMR applications to tackle future food fraud issues

pubblicato su: TRENDS IN FOOD SCIENCE & TECHNOLOGY - 2019

Sobolev Anatoly P., Thomas Freddy, Donarski James, Ingallina Cinzia, Circi Simone, Cesare Marincola Flaminia, Capitani Donatella, Mannina Luisa

A multi-methodological protocol to characterize PDO olive oils

pubblicato su: METABOLITES - 2018

Circi Simone, Ingallina Cinzia, Vista Silvia, Capitani Donatella, Di Vecchia Andrea, Leonardi Genesio, D’Achille Giovanni, Centauri Luigi, Camin Federica, Mannina Luisa

Selenotriapine - an isostere of the most studied thiosemicarbazone with pronounced pro-apoptotic activity, low toxicity and ability to challenge phenotype reprogramming of 3-D mammary adenocarcinoma tumors

pubblicato su: ARABIAN JOURNAL OF CHEMISTRY - 2020

Filipović N. R., Bjelogrlić S. K., Pelliccia S., Jovanović V. B., Kojić M., Senćanski M., La Regina G., Silvestri R., Muller C. D., Todorović T. R.

Discovery of new 1,1'-biphenyl-4-sulfonamides as selective subnanomolar human carbonic anhydrase II inhibitors

pubblicato su: ACS MEDICINAL CHEMISTRY LETTERS - 2020

La Regina G., Puxeddu M., Nalli M., Vullo D., Gratteri P., Supuran C. T., Nocentini A., Silvestri R.

Bax activation blocks self-renewal and induces apoptosis of human glioblastoma stem cells

pubblicato su: ACS CHEMICAL NEUROSCIENCE - 2018

Daniele S., Pietrobono D., Costa B., Giustiniano M., La Pietra V., Giacomelli C., LA REGINA Giuseppe, Silvestri Romano, Taliani S., Trincavelli M. L., Da Settimo F., Novellino E., Martini C., Marinelli L.

A negative allosteric modulator of WNT receptor frizzled 4 switches into an allosteric agonist

pubblicato su: BIOCHEMISTRY - 2018

Riccio G., Bottone S., La Regina G., Badolati N., Passacantilli S., Rossi G. B., Accardo A., Dentice M., Silvestri R., Novellino E., Stornaiuolo M.

DOACs: aspetti chimico-farmaceutici e tossicologici

pubblicato su: Anticoagulazione senza rischi - 2018

La Regina G.

New inhibitors of tubulin polymerization inspired by nature

pubblicato su: Pharma/Natural Products: Tecniche analitiche e nuove tendenze nel mondo dei prodotti naturali - 2018

La Regina G.

Sirtuin modulators: where are we now? A review of patents from 2015 to 2019

pubblicato su: EXPERT OPINION ON THERAPEUTIC PATENTS - 2020

Mautone Nicola, Zwergel Clemens, Mai Antonello, Rotili Dante

From parp1 to tnks2 Inhibition: a structure-based approach

pubblicato su: ACS MEDICINAL CHEMISTRY LETTERS - 2020

Tomassi Stefano, Pfahler Julian, Mautone Nicola, Rovere Annarita, Esposito Chiara, Passeri Daniela, Pellicciari Roberto, Novellino Ettore, Pannek Martin, Steegborn Clemens, Paiardini Alessandro, Mai Antonello, Rotili Dante

A closer look into NADPH oxidase inhibitors: validation and insight into their mechanism of action

pubblicato su: REDOX BIOLOGY - 2020

Reis J., Massari M., Marchese S., Ceccon M., Aalbers F. S., Corana F., Valente S., Mai A., Magnani F., Mattevi A.

Altered mitochondrial function in cells carrying a premutation or unmethylated full mutation of the FMR1 gene

pubblicato su: HUMAN GENETICS - 2020

Nobile V., Palumbo F., Lanni S., Ghisio V., Vitali A., Castagnola M., Marzano V., Maulucci G., De Angelis C., De Spirito M., Pacini L., D'Andrea L., Ragno R., Stazi G., Valente S., Mai A., Chiurazzi P., Genuardi M., Neri G., Tabolacci E.

Discovery of the first human arylsulfatase a reversible inhibitor impairing mouse oocyte fertilization

pubblicato su: ACS CHEMICAL BIOLOGY - 2020

Caroselli Silvia, Zwergel Clemens, Pirolli Adele, Sabatino Manuela, Xu Zhanjie, Kirsch Gilbert, Mai Antonello, Colotti Gianni, Altieri Fabio, Canipari Rita, Valente Sergio, Ragno Rino

Identification of Inhibitors to trypanosoma cruzi sirtuins based on compounds developed to human enzymes

pubblicato su: INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES - 2020

Matutino Bastos Tanira, Botelho Pereira Soares Milena, Haddad Franco Caio, Alcântara Laura, Antonini Lorenzo, Sabatino Manuela, Mautone Nicola, Holanda Freitas-Junior Lucio, Moraes Carolina Borsoi, Ragno Rino, Rotili Dante, Schenkman Sergio, Mai Antonello, Silvio Moretti Nilmar

The pan-sirtuin inhibitor MC2494 regulates mitochondrial function in a leukemia cell line

pubblicato su: FRONTIERS IN ONCOLOGY - 2020

Carafa Vincenzo, Russo Rosita, Della Torre Laura, Cuomo Francesca, Dell'Aversana Carmela, Sarno Federica, Sgueglia Giulia, Di Donato Marzia, Rotili Dante, Mai Antonello, Nebbioso Angela, Cobellis Gilda, Chambery Angela, Altucci Lucia

Sirt4: a multifaceted enzyme at the crossroads of mitochondrial metabolism and cancer

pubblicato su: FRONTIERS IN ONCOLOGY - 2020

Tomaselli D., Steegborn C., Mai A., Rotili D.

Detrimental effects of the 'bath salt' methylenedioxypyrovalerone on social play behavior in male rats

pubblicato su: NEUROPSYCHOPHARMACOLOGY - 2020

Schiavi Sara, Melancia Francesca, Carbone Emilia, Buzzelli Valeria, Manduca Antonia, Peinado Patricia Jiménez, Zwergel Clemens, Mai Antonello, Campolongo Patrizia, Vanderschuren Louk J M J, Trezza Viviana

The innovative potential of statins in cancer: new targets for new therapies

pubblicato su: FRONTIERS IN CHEMISTRY - 2020

Di Bello Elisabetta, Zwergel Clemens, Mai Antonello, Valente Sergio

Pharmacological inhibition of lysine-specific demethylase 1 (LSD1) induces global transcriptional deregulation and ultrastructural alterations that impair viability in Schistosoma mansoni

pubblicato su: PLOS NEGLECTED TROPICAL DISEASES - 2020

Coutinho Carneiro V., de Abreu da Silva I. C., Amaral M. S., Pereira A. S. A., Silveira G. O., Pires D. D. S., Verjovski-Almeida S., Dekker F. J., Rotili D., Mai A., Lopes-Torres E. J., Robaa D., Sippl W., Pierce R. J., Borrello M. T., Ganesan A., Lancelot J., Thiengo S., Fernandez M. A., Vicentino A. R. R., Mourao M. M., Coelho F. S., Fantappie M. R.

Acute and chronic neurobehavioral effects of the designer drug and bath salt constituent 3,4-methylenedioxypyrovalerone in the rat

pubblicato su: JOURNAL OF PSYCHOPHARMACOLOGY - 2019

Atehortua-Martinez Luisa Alessandra, Masniere Cyriaque, Campolongo Patrizia, Chasseigneaux Stéphanie, Callebert Jacques, Zwergel Clemens, Mai Antonello, Laplanche Jean-Louis, Chen Huixiong, Etheve-Quelquejeu Mélanie, Mégarbane Bruno, Benturquia Nadia

Effect of α-methoxy substitution on the anti-HIV activity of dihydropyrimidin-4(3 H)-ones

pubblicato su: JOURNAL OF MEDICINAL CHEMISTRY - 2019

Nawrozkij Maxim B., Forgione Mariantonietta, Yablokov Alexandre S., Lucidi Alessia, Tomaselli Daniela, Patsilinakos Alexandros, PANELLA CRISTINA, Hailu Gebremedhin S., Kirillov Ivan A., Badia Roger, Riveira-Munoz Eva, Crespan Emmanuele, Armijos Rivera Jorge I., Cirilli Roberto, Ragno Rino, Esté José A., Maga Giovanni, Mai Antonello, Rotili Dante

The emerging role of epigenetics in human autoimmune disorders

pubblicato su: CLINICAL EPIGENETICS - 2019

Mazzone Roberta, Zwergel Clemens, Artico Marco, Taurone Samanta, Ralli Massimo, Greco Antonio, Mai Antonello

Sirtuins as drug targets

pubblicato su: Epigenetic Drug Discovery - 2019

Zwergel Clemens, Rotili Dante, Valente Sergio, Mai Antonello