| Titolo |
Pubblicato in |
Anno |
| Bicyclic γ-amino acids as inhibitors of γ-aminobutyrate aminotransferase |
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY |
2016 |
| New Inhibitors of Dengue Virus Replication |
Abstract eBook |
2016 |
| New Inhibitors of indoleamine 2,3-dioxygenase 1: molecular modelling studies, synthesis and biological evaluation |
Abstract eBook |
2016 |
| New inhibitors of indoleamine 2,3-dioxygenase 1: molecular modeling studies, synthesis, and biological evaluation |
JOURNAL OF MEDICINAL CHEMISTRY |
2016 |
| Structure-based virtual screening to get new scaffold inhibitors of the Ser/Thr protein kinase PknB from Mycobacterium tuberculosis |
LETTERS IN DRUG DESIGN & DISCOVERY |
2016 |
| Focus on chirality of HIV-1 non-nucleoside reverse transcriptase inhibitors |
MOLECULES |
2016 |
| New 1-phenyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamides inhibit hepatitis C virus replication via suppression of cyclooxygenase-2 |
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY |
2015 |
| Structure-based lead optimization and biological evaluation of BAX direct activators as novel potential anticancer agents |
JOURNAL OF MEDICINAL CHEMISTRY |
2015 |
| Pharmacological folding chaperones act as allosteric ligands of Frizzled4 |
NATURE CHEMICAL BIOLOGY |
2015 |
| Kinetic characterization of 4,4'-biphenylsulfonamides as selective non-zinc binding MMP inhibitors |
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY |
2015 |
| Discovery of 1,1'-biiphenyl-4-sulfonamides as a new class of potent and selective carbonic anhydrase XIV inhibitors |
JOURNAL OF MEDICINAL CHEMISTRY |
2015 |
| Endogenous vs exogenous allosteric modulators in GPCRs: a dispute for shuttling CB1 among different membrane microenvironments |
SCIENTIFIC REPORTS |
2015 |
| New Indole Tubulin Assembly Inhibitors Cause Stable Arrest of Mitotic Progression, Enhanced Stimulation of Natural Killer Cell Cytotoxic Activity, and Repression of Hedgehog-Dependent Cancer |
JOURNAL OF MEDICINAL CHEMISTRY |
2015 |
| Poster: "In vivo selection of JARID histone demethylases inhibitors and their use to enlighten the biological role of these enzymes in yeast and mammalian cells with focus on transcriptional regulation” |
Abstracts of the 27th International Conference on Yeast Genetics and Molecular Biology |
2015 |
| New indole tubulin assembly inhibitors with stable arrest of mitotic progression, enhanced stimulation of natural killer cell cytotoxic activity and repression of Hedgehog-dependent cancer |
SIMCC2015 |
2015 |
| Synthesis of New Indoles with Potent Tubulin Polymerization Inhibiting Activity Including Hedgehog-Dependent Cancer and Enhanced Stimulation of NK Cell Cytotoxic Activity |
Abstract eBook |
2015 |
| New Pyrazolecarboxamides a s Anti-HCV Agents via Targeting Cyclooxygenase-2 |
Abstract eBook |
2015 |
| Drug Design and Synthesis of New Indolylarylsulfones as HIV-1 Non-nucleoside Reverse Transcriptase Inhibitors |
Abstract eBook |
2015 |
| In vitro characterisation of a pleconaril/pirodavir-like compound with potent activity against rhinoviruses |
VIROLOGY JOURNAL |
2015 |
| Antiproliferative and proapoptotic effects of a pyrrole containing arylthioindole in human Jurkat leukemia cell line and multidrug-resistant Jurkat/A4 cells |
CANCER BIOLOGY & THERAPY |
2015 |
