| Titolo |
Pubblicato in |
Anno |
| Anticancer activity of (S)-5-Chloro-3-((3,5-dimethylphenyl)sulfonyl)-N-(1-oxo-1-((pyridin-4-ylmethyl)amino)propan-2-yl)-1H-indole-2-carboxamide (RS4690), a new dishevelled 1 inhibitor |
CANCERS |
2022 |
| Single-run chemo- and enantio-selective high-performance liquid chromatography separation of tramadol and its principal metabolite, O-desmethyltramadol, using a chlorinated immobilized amylose-based chiral stationary phase under multimodal elution conditions |
SEPARATION SCIENCE PLUS |
2022 |
| Modulating undruggable targets to overcome cancer therapy resistance |
DRUG RESISTANCE UPDATES |
2022 |
| Exploring CCRL2 chemerin binding using accelerated molecular dynamics |
PROTEINS |
2022 |
| Discovery of novel human lactate dehydrogenase inhibitors: Structure-based virtual screening studies and biological assessment |
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY |
2022 |
| EFFICACY AND SAFETY OF A NOVEL FOOD SUPPLEMENT IN THE TREATMENT OF FUNCTIONAL DYSPEPSIA: A PILOT OPEN STUDY |
AGRO FOOD INDUSTRY HI-TECH |
2022 |
| Induction of Ferroptosis in Glioblastoma and Ovarian Cancers by a New Pyrrole Tubulin Assembly Inhibitor |
JOURNAL OF MEDICINAL CHEMISTRY |
2022 |
| Emerging Direct Targeting β-Catenin Agents |
MOLECULES |
2022 |
| Discovery of pyrrole derivatives for the treatment of glioblastoma and chronic myeloid leukemia |
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY |
2021 |
| CXCR4 antagonism sensitizes cancer cells to novel indole-based MDM2/4 inhibitors in glioblastoma multiforme |
EUROPEAN JOURNAL OF PHARMACOLOGY |
2021 |
| RS4651 suppresses lung fibroblast activation via the TGF-β1/SMAD signalling pathway |
EUROPEAN JOURNAL OF PHARMACOLOGY |
2021 |
| RS-5645 attenuates inflammatory cytokine storm induced by SARS-CoV-2 spike protein and LPS by modulating pulmonary microbiota |
INTERNATIONAL JOURNAL OF BIOLOGICAL SCIENCES |
2021 |
| Targeting PDZ domains as potential treatment for viral infections, neurodegeneration and cancer |
BIOLOGY DIRECT |
2021 |
| Discovery of a novel class of norovirus inhibitors with high barrier of resistance |
PHARMACEUTICALS |
2021 |
| Emerging therapeutic agents for colorectal cancer |
MOLECULES |
2021 |
| A METHOD TO MEASURE THE BARRIER EFFECT OF DRUGS AND ITS APPLICATION IN THE STUDY OF HYDROLYZED COLLAGEN |
AGRO FOOD INDUSTRY HI-TECH |
2021 |
| Selenotriapine - an isostere of the most studied thiosemicarbazone with pronounced pro-apoptotic activity, low toxicity and ability to challenge phenotype reprogramming of 3-D mammary adenocarcinoma tumors |
ARABIAN JOURNAL OF CHEMISTRY |
2020 |
| Design, synthesis and discovery of novel N,N'-carbazoyl-aryl-urea inhibitors of Zika NS5 methyltransferase and virus replication. |
CHEMMEDCHEM |
2020 |
| Discovery of new 1,1'-biphenyl-4-sulfonamides as selective subnanomolar human carbonic anhydrase II inhibitors |
ACS MEDICINAL CHEMISTRY LETTERS |
2020 |
| Structure-activity relationship studies and in vitro and in vivo anticancer activity of novel 3-aroyl-1,4-diarylpyrroles against solid tumors and hematological malignancies |
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY |
2020 |
