Pubblicazioni

Crystal structure of Leishmania mexicana cysteine protease B in complex with a high-affinity azadipeptide nitrile inhibitor

2020 - BIOORGANIC & MEDICINAL CHEMISTRY

Ribeiro, Jean F. R.; Cianni, Lorenzo; Li, Chan; Warwick, Thomas G.; De Vita, Daniela; Rosini, Fabiana; dos Reis Rocho, Fernanda; Martins, Felipe C. P.; Kenny, Peter W.; Lameira, Jeronimo; LeitÃ£o, Andrei; Emsley, Jonas; Montanari, Carlos A.

New thiopyrimidine-benzenesulfonamide conjugates as selective carbonic anhydrase II inhibitors: synthesis, in vitro biological evaluation, and molecular docking studies.

2020 - BIOORGANIC & MEDICINAL CHEMISTRY

Abdel-Mohsen, Ht; El Kerdawy, Am; Omar, Ma; Berrino, E; Abdelsamie, As; El Diwani, Hi; Supuran, Ct.

Synthesis and structure-activity relationship of nitrile-based cruzain inhibitors incorporating a trifluoroethylamine-based P2 amide replacement

2019 - BIOORGANIC & MEDICINAL CHEMISTRY

Gomes, Juliana C; Cianni, Lorenzo; Ribeiro, Jean; Dos Reis Rocho, Fernanda; da Costa Martins Silva, Samelyn; Batista, Pedro Henrique Jatai; Moraes, Carolina Borsoi; Franco, Caio Haddad; Freitas-Junior, Lucio H G; Kenny, Peter W; LeitÃ£o, Andrei; Burtoloso, Antonio C B; de Vita, Daniela; Montanari, Carlos A

Towards the development of activity-based probes for detection of lysine-specific demethylase-1 activity.

2017 - BIOORGANIC & MEDICINAL CHEMISTRY

Ourailidou, Me; Lenoci, A; Zwergel, Clemens; Rotili, Dante; Mai, Antonello; Dekker, F. j. 4.

3-Phenylalkyl-2H-chromenes and -chromans as novel rhinovirus infection inhibitors

2017 - BIOORGANIC & MEDICINAL CHEMISTRY

Conti, Cinzia; PROIETTI MONACO, Luca; Desideri, Nicoletta

Derivatives of caffeic acid, a natural antioxidant, as the basis for the discovery of novel nonpeptidic neurotrophic agents

2017 - BIOORGANIC & MEDICINAL CHEMISTRY

Moosavi, F.; Hosseini, R.; Rajaian, H.; Silva, T.; MagalhÃ£es e Silva, D.; Saso, L.; Edraki, N.; Miri, R.; Borges, F.; Firuzi, O.

A novel library of saccharin and acesulfame derivatives as potent and selective inhibitors of carbonic anhydrase IX and XII isoforms

2016 - BIOORGANIC & MEDICINAL CHEMISTRY

Carradori, Simone; Secci, Daniela; DE MONTE, Celeste; Mollica, Adriano; Ceruso, Mariangela; Akdemir, Atilla; Sobolev, Anatoly P; Codispoti, Rossella; DE COSMI, Federica; Guglielmi, Paolo; Supuran, Claudiu T.

Novel indole-based melatonin analogues: evaluation of antioxidant activity and protective effect against amyloid Î²-induced damage

2016 - BIOORGANIC & MEDICINAL CHEMISTRY

Gurer Orhan, H.; Karaaslan, C.; Ozcan, S.; Firuzi, O.; Tavakkoli, M.; Saso, Luciano; Suzen, S.

New trans dichloro (triphenylphosphine)platinum(II) complexes containing N-(butyl),N-(arylmethyl)amino ligands: Synthesis, cytotoxicity and mechanism of action

2016 - BIOORGANIC & MEDICINAL CHEMISTRY

Dalla Via, Lisa; GarcÃa ArgÃ¡ez, AÃda Nelly; Agostinelli, Enzo; Belli Dell'Amico, Daniela; Labella, Luca; Samaritani, Simona

Carbon nanotubes supported tyrosinase in the synthesis of lipophilic hydroxytyrosol and dihydrocaffeoyl catechols with antiviral activity against DNA and RNA viruses.

2015 - BIOORGANIC & MEDICINAL CHEMISTRY

Botta, G; Bizzarri, Bm; Garozzo, A; Timpanaro, Rossella; Bisignano, Benedetta; Amatore, Donatella; Palamara, ANNA TERESA; Nencioni, Lucia; Saladino, R.