Pubblicazioni

Structure-guided approach identifies a novel class of HIV-1 ribonuclease H inhibitors: binding mode insights through magnesium complexation and site-directed mutagenesis studies

2018 - MEDCHEMCOMM

Poongavanam, Vasanthanathan; Corona, Angela; Steinmann, Casper; Scipione, Luigi; Grandi, Nicole; Pandolfi, Fabiana; Di Santo, Roberto; Costi, Roberta; Esposito, Francesca; Tramontano, Enzo; Kongsted, Jacob

(Chalcogen)semicarbazones and their cobalt complexes differentiate HL-60 myeloid leukaemia cells and are cytotoxic towards tumor cell lines

2017 - MEDCHEMCOMM

TodoroviÄ, Tamara R.; VukaÅ¡inoviÄ, Jelena; Portalone, Gustavo; Suleiman, Sherif; GligorijeviÄ, Nevenka; BjelogrliÄ, Snezana; JovanoviÄ, Katarina; RaduloviÄ, SiniÅ¡a; AnÄelkoviÄ, Katarina; Cassar, Analisse; FilipoviÄ, Nenad R.; Schembri Wismayer, Pierre

Tetrahydroquinolinone derivatives as potent P-glycoprotein inhibitors: design, synthesis, biological evaluation and molecular docking analysis

2017 - MEDCHEMCOMM

Ranjbar, S.; Firuzi, O.; Edraki, N.; Shahraki, O.; Saso, L.; Khoshneviszadeh, M.; Miri, R.

Pro-apoptotic and pro-differentiation induction by 8-quinolinecarboxaldehyde selenosemicarbazone and its Co(III) complex in human cancer cell lines

2016 - MEDCHEMCOMM

FilipoviÄ, N. R.; BjelogrliÄ, S.; Portalone, G.; Pelliccia, S.; Silvestri, R.; KlisuriÄ, O.; SenÄanski, M.; StankoviÄ, D.; TodoroviÄ, T. R.; Muller, Christian D.

Histone demethylating agents as potential S-adenosyl-l-methionine-competitors

2016 - MEDCHEMCOMM

NavakauskienÄ, R.; Mori, Mattia; Christodoulou, M. S.; ZentelytÄ, A.; Botta, Bruno; Via, L. Dalla; Ricci, F.; Damia, G.; Passarella, D.; Zilio, C.; Martinet, N.

Erratum: Inclusion of new 5-fluorouracil amphiphilic derivatives in liposome formulation for cancer treatment (Med. Chem. Commun. (2015) 6 (1639-1642))

2016 - MEDCHEMCOMM

Petaccia, M.; Condello, M.; Giansanti, L.; La Bella, A.; Leonelli, F.; Meschini, S.; Gradella Villalva, D.; Pellegrini, E.; Ceccacci, F.; Galantini, L.; Mancini, G.

Pyrrole- and indole-containing tranylcypromine derivatives as novel lysine-specific demethylase 1 inhibitors active on cancer cells.

2015 - MEDCHEMCOMM

Veronica, Rodriguez; Valente, Sergio; Stefano, Rovida; Rotili, Dante; Stazi, Giulia; Lucidi, Alessia; Giuseppe, Ciossani; Andrea, Mattevi; Oronza A., Botrugno; Paola, Dessanti; Ciro, Mercurio; Paola, Vianello; Saverio, Minucci; Mario, Varasi; Mai, Antonello

Inclusion of new 5-fluorouracil amphiphilic derivatives in liposome formulation for cancer treatment

2015 - MEDCHEMCOMM

Petaccia, M.; Condello, M.; Giansanti, L.; LA BELLA, Angela; Leonelli, Francesca; Meschini, S.; GRADELLA VILLALVA, Denise; Pellegrini, E.; Ceccacci, Francesca; Galantini, Luciano; Mancini, G.

The first potent diphenyl phosphonate KLK4 inhibitors with unexpected binding kinetics

2015 - MEDCHEMCOMM

van Soom, Jeroen; Cuzzucoli Crucitti, Giuliana; Gladysz, Rafaela; van der Veken, Pieter; Di Santo, Roberto; Stuyver, Ingmar; Buck, Victoria; Lambeir, Anne-Marie; Magdolen, Viktor; Joossens, Jurgen; Augustyns, Koen