Pubblicazioni

Emerging Therapeutic Potential of SIRT6 Modulators

2021 - JOURNAL OF MEDICINAL CHEMISTRY

Fiorentino, F.; Mai, A.; Rotili, D.

In silico and in vitro analysis of major cannabis-derived compounds as fatty acid amide hydrolase inhibitors

2021 - MOLECULES

Criscuolo, E.; De Sciscio, M. L.; Fezza, F.; Maccarrone, M.

Modification of the anabaseine pyridine nucleus allows achieving binding and functional selectivity for the Î±3Î²4 nicotinic acetylcholine receptor subtype

2016 - EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Matera, Carlo; Quadri, Marta; Sciaccaluga, Miriam; PomÃ¨, Diego Yuri; Fasoli, Francesca; De Amici, Marco; Fucile, Sergio; Gotti, Cecilia; Dallanoce, Clelia; Grazioso, Giovanni

Potent dual inhibitors of Plasmodium falciparum M1 and M17 aminopeptidases through optimization of S1 pocket interactions

2016 - EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Drinkwater, Nyssa; Vinh, Natalie B.; Mistry, Shailesh N.; Bamert, Rebecca S.; Ruggeri, Chiara; Holleran, John P.; Loganathan, Sasdekumar; Paiardini, Alessandro; Charman, Susan A.; Powell, Andrew K.; Avery, Vicky M.; Mcgowan, Sheena; Scammells, Peter J.

Inhibition of human monoamine oxidase: biological and molecular modeling studies on selected natural flavonoids

2016 - JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY

Carradori, Simone; Gidaro, Maria Concetta; Petzer, AnÃ©l; Costa, GiosuÃ¨; Guglielmi, Paolo; Chimenti, Paola; Alcaro, Stefano; Petzer, Jacobus P.

Enzyme kinetics and inhibition of histone acetyltransferase KAT8

2015 - EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Wapenaar, Hannah; van der Wouden, Petra E; Groves, Matthew R; Rotili, Dante; Mai, Antonello; Dekker, Frank J.

Chemistry and pharmacology of a series of unichiral analogues of 2-(2-pyrrolidinyl)-1,4-benzodioxane, prolinol phenyl ether, and prolinol 3-pyridyl ether designed as Î±4Î²2-nicotinic acetylcholine receptor agonists

2015 - JOURNAL OF MEDICINAL CHEMISTRY

Bolchi, Cristiano; Valoti, Ermanno; Gotti, Cecilia; Fasoli, Francesca; Ruggeri, Paola; Fumagalli, Laura; Binda, Matteo; Mucchietto, Vanessa; Sciaccaluga, Miriam; Budriesi, Roberta; Fucile, Sergio; Pallavicini, Marco