Pubblicazioni

Vibrational circular dichroism (VCD) reveals subtle conformational aspects and intermolecular interactions in the carnitine family

2015 - CHIRALITY

Mazzeo, Giuseppe; Abbate, Sergio; Longhi, Giovanna; Castiglioni, Ettore; VILLANI, Claudio

Targeting the noradrenergic system in posttraumatic stress disorder. A systematic review and meta-analysis of prazosin trials

2015 - CURRENT DRUG TARGETS

de Berardis, Domenico; Marini, Stefano; Serroni, Nicola; Iasevoli, Felice; Tomasetti, Carmine; de Bartolomeis, Andrea; Mazza, Monica; Tempesta, Daniela; Valchera, Alessandro; Fornaro, Michele; Pompili, Maurizio; Sepede, Gianna; Vellante, Federica; Orsolini, Laura; Martinotti, Giovanni; Di Giannantonio, Massimo

Discovery of N-aryl-naphthylamines as in vitro inhibitors of the interaction between HIV integrase and the cofactor LEDGF/p75

2015 - EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Cuzzucoli Crucitti, G.; Pescatori, Luca; Messore, A. A; Madia, VALENTINA NOEMI; Pupo, Giovanni; Saccoliti, Francesco; Scipione, Luigi; Tortorella, Silvano; Di Leva, F. S; Cosconati, S; Novellino, E; Debyser, Z; Christ, F; Costi, Roberta; DI SANTO, Roberto

Exploring oxidovanadium(IV) complexes as YopH inhibitors: mechanism of action and modeling studies

2015 - ACS MEDICINAL CHEMISTRY LETTERS

Martins, Priscila G. A; Mori, Mattia; Chiaradia Delatorre, Louise D; Menegatti, Angela C. O; Mascarello, Alessandra; Botta, Bruno; BenÃtez, Julio; Gambino, Dinorah; Terenzi, HernÃ¡n

"Natural" relief of pregnancy-related symptoms and neonatal outcomes: above all do no harm

2015 - JOURNAL OF ETHNOPHARMACOLOGY

Trabace, Luigia; Tucci, Paolo; Ciuffreda, Lucia; Matteo, Maria; Fortunato, Francesca; Campolongo, Patrizia; Trezza, Viviana; Cuomo, Vincenzo

A facile palladium-catalyzed route to 2,5,7-trisubstituted indoles

2015 - TETRAHEDRON

Cacchi, Sandro; Fabrizi, Giancarlo; Goggiamani, Antonella; Iazzetti, Antonia; Verdiglione, Rosanna

Emerging approaches for histone deacetylase inhibitor drug discovery

2015 - EXPERT OPINION ON DRUG DISCOVERY

Zwergel, Clemens; Valente, Sergio; Jacob, Claus; Mai, Antonello

Differential effects of extracellular vesicles secreted by mesenchymal stem cells from different sources on glioblastoma cells

2015 - EXPERT OPINION ON BIOLOGICAL THERAPY

Del Fattore, Andrea; Luciano, Rosa; Saracino, Rossana; Battafarano, Giulia; Rizzo, Cristiano; Pascucci, Luisa; Alessandri, Giulio; Pessina, Augusto; Perrotta, Antonio; Fierabracci, Alessandra; Muraca, Maurizio

A novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach

2015 - JOURNAL OF MEDICINAL CHEMISTRY

Milite, Ciro; Feoli, Alessandra; Sasaki, Kazuki; La Pietra, Valeria; Balzano, Amodio Luca; Marinelli, Luciana; Mai, Antonello; Novellino, Ettore; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca

Chemistry and pharmacology of a series of unichiral analogues of 2-(2-pyrrolidinyl)-1,4-benzodioxane, prolinol phenyl ether, and prolinol 3-pyridyl ether designed as Î±4Î²2-nicotinic acetylcholine receptor agonists

2015 - JOURNAL OF MEDICINAL CHEMISTRY

Bolchi, Cristiano; Valoti, Ermanno; Gotti, Cecilia; Fasoli, Francesca; Ruggeri, Paola; Fumagalli, Laura; Binda, Matteo; Mucchietto, Vanessa; Sciaccaluga, Miriam; Budriesi, Roberta; Fucile, Sergio; Pallavicini, Marco

New amide derivatives of Probenecid as selective inhibitors of carbonic anhydrase IX and XII: Biological evaluation and molecular modelling studies

2015 - BIOORGANIC & MEDICINAL CHEMISTRY

Carradori, Simone; Mollica, Adriano; Ceruso, Mariangela; D'Ascenzio, Melissa; DE MONTE, Celeste; Chimenti, Paola; Sabia, Rocchina; Akdemir, Atilla; Supuran, Claudiu T.

Diastereomer Interconversion via Enolization: A Case Study

2015 - CHIRALITY

Renzetti, Andrea; Di Crescenzo, Antonello; Nie, Feilin; Bond, Andrew D.; GÃ©rard, StÃ©phane; Sapi, Janos; Fontana, Antonella; Villani, Claudio

Synthesis, biological evaluation and docking analysis of a new series of methylsulfonyl and sulfamoyl acetamides and ethyl acetates as potent COX-2 inhibitors

2015 - BIOORGANIC & MEDICINAL CHEMISTRY

Consalvi, Sara; Alfonso, Salvatore; Di Capua, Angela; Poce, Giovanna; Pirolli, Adele; Sabatino, Manuela; Ragno, Rino; Anzini, Maurizio; Sartini, Stefania; La Motta, Concettina; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Biava, Mariangela

Efficacy of trabectedin in advanced soft tissue sarcoma: Beyond lipo- and leiomyosarcoma

2015 - DRUG DESIGN, DEVELOPMENT AND THERAPY

DE SANCTIS, Rita; Marrari, Andrea; Marchetti, Silvia; Mussi, Chiara; Balzarini, Luca; Lutman, Fabio Romano; Daolio, Primo; Bastoni, Stefano; Bertuzzi, Alexia Francesca; Quagliuolo, Vittorio; Santoro, Armando