Pubblicazioni

New 1-phenyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamides inhibit hepatitis C virus replication via suppression of cyclooxygenase-2

2015 - EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Manvar, D.; Pelliccia, S.; La Regina, G.; Famiglini, V.; Coluccia, A.; Ruggieri, A.; Anticoli, S.; Lee, J. -C.; Basu, A.; Cevik, O.; Nencioni, L.; Palamara, A. T.; Zamperini, C.; Botta, M.; Neyts, J.; Leyssen, P.; Kaushik-Basu, N.; Silvestri, R.

Synthesis and structure-activity relationship of new cytotoxic agents targeting human glutathione-S-transferases.

2015 - EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Rotili, Dante; De Luca, A; Tarantino, D; Pezzola, S; Forgione, Mariantonietta; Morozzo Della Rocca, B; Falconi, M; Mai, Antonello; Caccuri, A. M.

Pure enantiomers of benzoylamino-tranylcypromine: LSD1 inhibition, gene modulation in human leukemia cells and effects on clonogenic potential of murine promyelocytic blasts

2015 - EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

VALENTE, Sergio; Veronica, Rodriguez; Mercurio, Ciro; Vianello, Paola; Saponara, Bruna; Cirilli, Roberto; Ciossani, Giuseppe; LABELLA, DONATELLA; MARROCCO, BIAGINA; Monaldi, Daria; RUOPPOLO, Giovanni; Tilset, Mats; Botrugno, Oronza A.; Dessanti, Paola; Minucci, Saverio; MATTEVI, ANDREA; Varasi, Mario; MAI, Antonello

Bifunctional compounds targeting both D2 and non-Î±7 nACh receptors: design, synthesis and pharmacological characterization

2015 - EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Matera, Carlo; Pucci, Luca; Fiorentini, Chiara; Fucile, Sergio; Missale, Cristina; Grazioso, Giovanni; Clementi, Francesco; Zoli, Michele; De Amici, Marco; Gotti, Cecilia; Dallanoce, Clelia

Synthesis and pharmacological screening of a large library of 1,3,4-thiadiazolines as innovative therapeutic tools for the treatment of prostate cancer and melanoma

2015 - EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

De Monte, Celeste; Carradori, Simone; Secci, Daniela; D'Ascenzio, Melissa; Guglielmi, Paolo; Mollica, Adriano; Morrone, Stefania; Scarpa, Susanna; Agliano', Anna Maria; Giantulli, Sabrina; Silvestri, Ida

Discovery of N-aryl-naphthylamines as in vitro inhibitors of the interaction between HIV integrase and the cofactor LEDGF/p75

2015 - EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Cuzzucoli Crucitti, G.; Pescatori, Luca; Messore, A. A; Madia, VALENTINA NOEMI; Pupo, Giovanni; Saccoliti, Francesco; Scipione, Luigi; Tortorella, Silvano; Di Leva, F. S; Cosconati, S; Novellino, E; Debyser, Z; Christ, F; Costi, Roberta; DI SANTO, Roberto

Enzyme kinetics and inhibition of histone acetyltransferase KAT8

2015 - EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Wapenaar, Hannah; van der Wouden, Petra E; Groves, Matthew R; Rotili, Dante; Mai, Antonello; Dekker, Frank J.