Pubblicazioni

TRPA1 channels as targets for resveratrol and related stilbenoids

2016 - BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Nalli, Marianna; Ortar, Giorgio; Moriello, Aniello Schiano; Morera, Enrico; Di Marzo, Vincenzo; De Petrocellis, Luciano

Synthesis and biological evaluation of fluorinated 1,5-diarylpyrrole-3-alkoxyethyl ether derivatives as selective COX-2 inhibitors endowed with anti-inflammatory activity

2016 - EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Di Capua, Angela; Sticozzi, Claudia; Brogi, Simone; Brindisi, Margherita; Cappelli, Andrea; Sautebin, Lidia; Rossi, Antonietta; Pace, Simona; Ghelardini, Carla; Di Cesare Mannelli, Lorenzo; Valacchi, Giuseppe; Giorgi, Gianluca; Giordani, Antonio; Poce, Giovanna; Biava, Mariangela; Anzini, Maurizio

(E)-3-Heteroarylidenechroman-4-ones as potent and selective monoamine oxidase-B inhibitors

2016 - EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Desideri, Nicoletta; PROIETTI MONACO, Luca; Fioravanti, Rossella; Biava, Mariangela; YÃ¡Ã±ez, Matilde; Alcaro, Stefano; Ortuso, Francesco

VP1 crystal structure-guided exploration and optimization of 4,5-dimethoxybenzene-based inhibitors of rhinovirus 14 infection

2016 - EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Da Costa, LaurÃ¨ne; Roche, Manon; Scheers, Els; Coluccia, Antonio; Neyts, Johan; Terme, Thierry; Leyssen, Pieter; Silvestri, Romano; Vanelle, Patrice

Bicyclic Î³-amino acids as inhibitors of Î³-aminobutyrate aminotransferase

2016 - JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Pinto, Andrea; Tamborini, Lucia; Pennacchietti, Eugenia; Coluccia, Antonio; Silvestri, Romano; Cullia, Gregorio; De Micheli, Carlo; Conti, Paola; DE BIASE, Daniela

High-performance liquid chromatographic resolution of neutral and cationic hetero[6]helicenes

2016 - CHIRALITY

Labrador, Geraldine M.; Bosson, Johann; Breitbach, Zachary S.; Lim, Yeeun; Francotte, Eric R.; Sabia, Rocchina; Villani, Claudio; Armstrong, Daniel W.; Lacour, JÃ©rÃ´me

Extraction of bioactive polyphenols with high antioxidant activity from bilberry (Vaccinium myrtillus L.) processing waste

2016 - ORIENTAL JOURNAL OF CHEMISTRY

Fidaleo, Marcello; Lavecchia, Roberto; Zuorro, Antonio

Determination of different recreational drugs in sweat by headspace solid-phase microextraction gas chromatography mass spectrometry (HS-SPME GC/MS): application to drugged drivers

2016 - JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS

Gentili, Stefano; Mortali, Claudia; Mastrobattista, Luisa; Berretta, Paolo; Zaami, Simona

The novel antipsychotic cariprazine (RGH-188). State-of-the-art in the treatment of psychiatric disorders

2016 - CURRENT PHARMACEUTICAL DESIGN

De Berardis, Domenico; Orsolini, Laura; Iasevoli, Felice; Prinzivalli, Emiliano; De Bartolomeis, Andrea; Serroni, Nicola; Mazza, Monica; Valchera, Alessandro; Fornaro, Michele; Vecchiotti, Roberta; Carano, Alessandro; Sepede, Gianna; Vellante, Federica; Matarazzo, Ilaria; Pompili, Maurizio; Perna, Giampaolo; Conti, Chiara; GarcÃa, Cristina Segura; Martinotti, Giovanni; Di Giannantonio, Massimo

Modification of the anabaseine pyridine nucleus allows achieving binding and functional selectivity for the Î±3Î²4 nicotinic acetylcholine receptor subtype

2016 - EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Matera, Carlo; Quadri, Marta; Sciaccaluga, Miriam; PomÃ¨, Diego Yuri; Fasoli, Francesca; De Amici, Marco; Fucile, Sergio; Gotti, Cecilia; Dallanoce, Clelia; Grazioso, Giovanni

Evaluation of the analgesic effect of 4-anilidopiperidine scaffold containing ureas and carbamates

2016 - JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Monti, Ludovica; Stefanucci, Azzurra; Pieretti, Stefano; Marzoli, Francesca; Fidanza, Lorenzo; Mollica, Adriano; Mirzaie, Sako; Carradori, Simone; Petrocellis, Luciano De; Moriello, Aniello Schiano; Benyhe, Sa Ìndor; Ferenc Za, Ìdor; Szucs, Edina; Ferenc O., Ìtvos; Erdei, Anna I.; Samavati, Reza; Szabolcs Dvora, Ìcsko; Csaba To Ìmbo, Ìly; Novellino, Ettore

Purification, conformational analysis, and properties of a family of tigerinin peptides from skin secretions of the crowned bullfrog hoplobatrachus occipitalis

2016 - JOURNAL OF NATURAL PRODUCTS

Mclaughlin, Christopher M.; Lampis, Sandrina; Mechkarska, Milena; Coquet, Laurent; Jouenne, Thierry; King, Jay D.; Mangoni, Maria Luisa; Lukic, Miodrag L.; Scorciapino, Mariano A.; Conlon, J. Michael

MC1568 inhibits HDAC6/8 activity and influenza A virus replication in lung epithelial cells: Role of Hsp90 acetylation

2016 - FUTURE MEDICINAL CHEMISTRY

Panella, Simona; Marcocci, Maria Elena; Celestino, Ignacio; Valente, Sergio; Zwergel, Clemens; Li Puma, Domenica Donatella; Nencioni, Lucia; Mai, Antonello; Palamara, ANNA TERESA; Simonetti, Giovanna

Cathepsin D as a therapeutic target in Alzheimerâs disease

2016 - EXPERT OPINION ON THERAPEUTIC TARGETS

Di Domenico, Fabio; Tramutola, Antonella; Perluigi, Marzia

Potent dual inhibitors of Plasmodium falciparum M1 and M17 aminopeptidases through optimization of S1 pocket interactions

2016 - EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Drinkwater, Nyssa; Vinh, Natalie B.; Mistry, Shailesh N.; Bamert, Rebecca S.; Ruggeri, Chiara; Holleran, John P.; Loganathan, Sasdekumar; Paiardini, Alessandro; Charman, Susan A.; Powell, Andrew K.; Avery, Vicky M.; Mcgowan, Sheena; Scammells, Peter J.

Mycobacterium tuberculosis-secreted tyrosine phosphatases as targets against tuberculosis: exploring natural sources in searching for new drugs

2016 - CURRENT PHARMACEUTICAL DESIGN

Mascarello, Alessandra; Chiaradia Delatorre, Louise Domeneghini; Mori, Mattia; Terenzi, HernÃ¡n; Botta, Bruno

Achiral dye/surfactant heteroaggregates for chiral sensing of phosphocholines

2016 - CHIRALITY

Ceccacci, Francesca; Scipioni, Anita; Altieri, Barbara; Giansanti, Luisa; Mancini, Giovanna

MmpL3 inhibitors: diverse chemical scaffolds inhibit the same target

2016 - MINI-REVIEWS IN MEDICINAL CHEMISTRY

Poce, Giovanna; Consalvi, Sara; Biava, Mariangela