Pubblicazioni

Inhibition of Leishmania infantum trypanothione reductase by diaryl sulfide derivatives

2017 - JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Saccoliti, Francesco; Angiulli, Gabriella; Pupo, Giovanni; Pescatori, Luca; Madia, VALENTINA NOEMI; Messore, Antonella; Colotti, Gianni; Fiorillo, Annarita; Scipione, Luigi; Gramiccia, Marina; Di Muccio, Trentina; DI SANTO, Roberto; Costi, Roberta; Ilari, Andrea

A new nitrobenzoxadiazole-based GSTP1-1 inhibitor with a previously unheard of mechanism of action and high stability.

2017 - JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Fulci, C; Rotili, Dante; De Luca, A; Stella, L; Morozzo Della Rocca, B; Forgione, M; Di Paolo, V; Mai, Antonello; Falconi, M; Quintieri, L; Caccuri, Am; 7, .

pH-sensitive niosomes: effects on cytotoxicity and on inflammation and pain in murine models

2017 - JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Rinaldi, Federica; Del Favero, Elena; Rondelli, Valeria; Pieretti, Stefano; Bogni, Alessia; Ponti, Jessica; Rossi, François; Di Marzio, Luisa; Paolino, Donatella; Marianecci, Carlotta; Carafa, Maria

Exploring the first Rimonabant analog-​opioid peptide hybrid compound, as bivalent ligand for CB1 and opioid receptors

2017 - JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Mollica, Adriano; Pelliccia, Sveva; Famiglini, Valeria; Stefanucci, Azzurra; Macedonio, Giorgia; Chiavaroli, Annalisa; Orlando, Giustino; Brunetti, Luigi; Ferrante, Claudio; Pieretti, Stefano; Novellino, Ettore; Benyhe, Sandor; Zador, Ferenc; Erdei, Anna; Szucs, Edina; Samavati, Reza; Dvrorasko, Szalbolch; Tomboly, Csaba; Ragno, Rino; Patsilinakos, Alexandros; Silvestri, Romano

Synthesis, biological evaluation and molecular modeling studies on novel quinonoid inhibitors of CDC25 phosphatases

2017 - JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Evain Bana, Emilie; Schiavo, Lucie; Bour, Christophe; Lanfranchi, Don Antoine; Berardozzi, Simone; Ghirga, Francesca; Bagrel, Denyse; Botta, Bruno; Hanquet, Gilles; Mori, Mattia

Inhibition of the α-carbonic anhydrase from Vibrio cholerae with amides and sulfonamides incorporating imidazole moieties

2017 - JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
DE VITA, Daniela; Angeli, Andrea; Pandolfi, Fabiana; Bortolami, Martina; Costi, Roberta; DI SANTO, Roberto; Suffredini, Elisabetta; Ceruso, Mariangela; Del Prete, Sonia; Capasso, Clemente; Scipione, Luigi; Supuran, Claudiu T.

Synthesis and biological evaluation of anti-Toxoplasma gondii activity of a novel scaffold of thiazolidinone derivatives

2017 - JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Carradori, Simone; Secci, Daniela; Bizzarri, Bruna; Chimenti, Paola; DE MONTE, Celeste; Guglielmi, Paolo; Campestre, Cristina; Rivanera, Daniela; Bordón, Claudia; Jones Brando, Lorraine

Open saccharin-based secondary sulfonamides as potent and selective inhibitors of cancer-related carbonic anhydrase IX and XII isoforms

2017 - JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
D'Ascenzio, M.; Guglielmi, P.; Carradori, S.; Secci, D.; Florio, R.; Mollica, A.; Ceruso, M.; Akdemir, A.; Sobolev, A. P.; Supuran, C. T.

Neem oil nanoemulsions: characterisation and antioxidant activity

2017 - JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Rinaldi, Federica; Hanieh, PATRIZIA NADIA; Longhi, Catia; Carradori, Simone; Secci, Daniela; Zengin, Gokhan; Grazia Ammendolia, Maria; Mattia, Elena; Del Favero, Elena; Marianecci, Carlotta; Carafa, Maria

Inhibition of dengue virus replication by novel inhibitors of RNA-dependent RNA polymerase and protease activities

2017 - JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Pelliccia, S.; Wub, Y. H.; Coluccia, A.; La Regina, G.; Tseng, C. K.; Famiglini, V.; Masci, D.; Hiscott, J.; Lee, J. C.; Silvestri, R.

Expression of heterologous oxalate decarboxylase in HEK293 cells confers protection against oxalate induced oxidative stress as a therapeutic approach for calcium oxalate stone disease

2017 - JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Albert, A.; Tiwari, V.; Paul, E.; Ganesan, D.; Ayyavu, M.; Kujur, R.; Ponnusamy, S.; Shanmugam, K.; Saso, L.; Govindan Sadasivam, S.

Disulfiram moderately restores impaired hepatic redox status of rats subchronically exposed to cadmium

2017 - JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Begic, A.; Djuric, A.; Ninkovic, M.; Stevanovic, I.; Djurdjevic, D.; Pavlovic, M.; Jelic, K.; Pantelic, A.; Zebic, G.; Dejanovic, B.; Stanojevic, I.; Vojvodic, D.; Milosavljevic, P.; Djukic, M.; Saso, L.

Analysis of imidazoles and triazoles in biological samples after MicroExtraction by packed sorbent

2017 - JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Campestre, Cristina; Locatelli, Marcello; Guglielmi, Paolo; De Luca, Elisa; Bellagamba, Giuseppe; Menta, Sergio; Zengin, Gokhan; Celia, Christian; Di Marzio, Luisa; Carradori, Simone

Metabolite profiling of ascidian Styela plicata using LC–MS with multivariate statistical analysis and their antitumor activity

2017 - JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Palanisamy, S. K.; Trisciuoglio, D.; Zwergel, C.; Del Bufalo, D.; Mai, A.

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